EFFECT OF A NEW POTENT H2-RECEPTOR ANTAGONIST 3[[[2-[(DIAMINOMETHYLENE)AMINO]-4-THIAZOLYL]METHYL]THIO]-N-2-SULFAMOYLPROPIONAMIDINE (YM-11170) ON GASTRIC-MUCOSAL HISTAMINE-SENSITIVE ADENYLATE-CYCLASE FROM GUINEA-PIG

被引:36
作者
HARADA, M [1 ]
TERAI, M [1 ]
MAENO, H [1 ]
机构
[1] YAMANOUCHI PHARMACEUT CO LTD,DEPT BIOCHEM,CENT RES LABS,TOKYO 174,JAPAN
关键词
D O I
10.1016/0006-2952(83)90339-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1635 / 1640
页数:6
相关论文
共 31 条
[1]   STIMULATION OF ADENYLATE-CYCLASE OF GUINEA-PIG GASTRIC-MUCOSA BY HISTAMINE, SODIUM-FLUORIDE AND 5'-GUANYLYLIMIDODIPHOSPHATE AND INHIBITION BY HISTAMINE H1-RECEPTOR AND H2-RECEPTOR ANTAGONISTS INVITRO [J].
ANTTILA, P ;
LUCKE, C ;
WESTERMANN, E .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1976, 296 (01) :31-36
[2]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[3]  
BROWN BL, 1972, ADV CYCL NUCL RES<D>, V2, P25
[4]  
BYLUND DB, 1976, MOL PHARMACOL, V12, P568
[5]  
CHERET AM, 1981, MOL PHARMACOL, V20, P326
[6]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[7]  
DIXON M, 1979, ENZYMES, P60
[8]  
DOUSA TP, 1977, GASTROENTEROLOGY, V73, P904
[9]   EFFECT OF HISTAMINE AND ITS METHYL-DERIVATIVES ON CYCLIC-AMP METABOLISM IN GASTRIC-MUCOSA AND ITS BLOCKADE BY AN H2 RECEPTOR ANTAGONIST [J].
DOUSA, TP ;
CODE, CF .
JOURNAL OF CLINICAL INVESTIGATION, 1974, 53 (01) :334-337
[10]   EFFECT OF HISTAMINE ON CANINE GASTRIC MUCOSAL ADENYLATE-CYCLASE [J].
DOZOIS, RR ;
WOLLIN, A ;
RETTMANN, RD ;
DOUSA, TP .
AMERICAN JOURNAL OF PHYSIOLOGY, 1977, 232 (01) :E35-E38