ELECTROCHEMICAL AND ANTIBACTERIAL BEHAVIOR OF DERIVATIVES OF (1S, 2S) - 2 AMINO- 1- (4-NITROPHENYL) - PROPANE-1,3-DIOL

被引:0
|
作者
Cristea, Cecilia [1 ]
Voiculescu, G. [2 ]
Jitaru, Maria [2 ]
Moinet, C. [3 ]
机构
[1] Univ Med & Pharm Iuliu Hatieganu, Fac Pharm, Dept Chim Analyt, 4 Rue Pasteur, Cluj Napoca 400349, Romania
[2] Univ Babes Bolyai Cluj Napoca, Lab Assoc Francophone, Cluj Napoca 400028, Romania
[3] Univ Rennes 1, Inst Chim, Lab Electrochim & Organometall, F-35042 Rennes, France
关键词
electrosynthesis; hydroxylamines; nitrosoderivatives; redox cell;
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
Derivatives of (1S, 2S)-2-amino-1-(4-nitrophenyl)propane-1,3-diol were studied because of their potential biological activity. Using the electrogenerated intermediates (hydroxylamine and nitroso derivatives) N-sulphonylphenylhydroxylamines and benzoxazine diones were obtained with good yields. Their antibacterial activity was investigated on several gram-negative and gram-positive bacilli by two techniques: broth-dilution method and agar-dilution method.
引用
收藏
页码:209 / 216
页数:8
相关论文
共 50 条
  • [1] Electrosynthesis of nitroso compounds from (1S, 2S)-2-amino-l-(4-nitrophenyl)-propane-1,3-diol derivatives
    C. V. Cristea
    C. Moinet
    M. Jitaru
    I. C. Popescu
    Journal of Applied Electrochemistry, 2005, 35 : 851 - 855
  • [2] Electrosynthesis of nitroso compounds from (1S,2S)-2-amino-l-(4-nitrophenyl)-propane-1,3-diol derivatives
    Cristea, CV
    Moinet, C
    Jitaru, M
    Popescu, IC
    JOURNAL OF APPLIED ELECTROCHEMISTRY, 2005, 35 (09) : 851 - 855
  • [3] RESOLUTION OF THE ENANTIOMERS OF (S,R)-1,1'-BI-2,2'-NAPHTHYLHYDROGENPHOSPHATE BY (1R,2R)-2-AMINO-1-(4-NITROPHENYL)-PROPANE-1,3-DIOL AND (1S,2S)-2-AMINO-1-(4-NITROPHENYL)-PROPANE-1,3-DIOL
    WERNER, W
    TRESSELT, D
    IHN, W
    ZIEBELL, G
    JOURNAL FUR PRAKTISCHE CHEMIE, 1987, 329 (06): : 1031 - 1037
  • [4] Electroreduction of (1S,2S)-2-amino-1-(4-nitrophenyl)-propane-1,3-diol derivatives. Behaviour of electrogenerated species and applications to organic synthesis
    C.V. Cristea
    C. Moinet
    M. JITARU
    M. Darabantu
    Journal of Applied Electrochemistry, 2005, 35 : 845 - 849
  • [5] Electroreduction of (1S,2S)-2-amino-1-(4-nitrophenyl)-propane-1,3-diol derivatives.: Behaviour of electrogenerated species and applications to organic synthesis
    Cristea, CV
    Moinet, C
    Jitaru, M
    Darabantu, M
    JOURNAL OF APPLIED ELECTROCHEMISTRY, 2005, 35 (09) : 845 - 849
  • [6] (1S*,2S*)-(+)-2-amino-1-[4-(methylsulfanyl)phenyl]propane-1,3-diol
    Samas, B
    Macikenas, D
    Blackburn, AC
    ACTA CRYSTALLOGRAPHICA SECTION E-CRYSTALLOGRAPHIC COMMUNICATIONS, 2005, 61 : O2793 - O2794
  • [7] Novel N-modified glycines based on a (1S,2S)-2-amino-1-(4-nitrophenyl) propane-1,3-diol skeleton: 1,3-dioxanes and tripodands
    Moldovan, Oana
    Albert, Katalin
    Nagy, Iulia
    Morar, Cristina
    Sacalis, Carmen
    Darabantu, Mircea
    TETRAHEDRON LETTERS, 2016, 57 (51) : 5808 - 5811
  • [8] POLAROGRAPHY OF D-THREO-1-[4-NITROPHENYL]-2-[AZIDOACETAMIDO]PROPANE-1,3-DIOL, AZIDAMPHENICOL
    PFLEGEL, P
    WAGNER, G
    PHARMAZIE, 1972, 27 (03): : 148 - &
  • [9] Synthesis and antimicrobial activity of urea derivatives of (1S,2S)-2-AMINO-1-(4-nitrophenyl)-1,3-propanediol
    M. Madesclaire
    S. Kh. Sharipova
    A. V. Lyamin
    A. A. Osipova
    E. A. Botkin
    Yu. V. Zaitseva
    V. P. Zaitsev
    Pharmaceutical Chemistry Journal, 2012, 45 : 668 - 670
  • [10] SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF UREA DERIVATIVES OF (1S,2S)-2-AMINO-1-(4-NITROPHENYL)-1,3-PROPANEDIOL
    Madesclaire, M.
    Sharipova, S. Kh.
    Lyamin, A. V.
    Osipova, A. A.
    Botkin, E. A.
    Zaitseva, Yu. V.
    Zaitsev, V. P.
    PHARMACEUTICAL CHEMISTRY JOURNAL, 2012, 45 (11) : 668 - 670