ANALGESIC ACTIVITY OF ENKEPHALINS FOLLOWING INTRACEREBRAL ADMINISTRATION IN RAT

被引:43
作者
MALICK, JB [1 ]
GOLDSTEIN, JM [1 ]
机构
[1] STUART PHARMACEUT,DEPT BIOMED RES,WILMINGTON,DE 19897
关键词
D O I
10.1016/0024-3205(77)90034-0
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:827 / 832
页数:6
相关论文
共 19 条
[1]   ANALGESIA INDUCED INVIVO BY CENTRAL ADMINISTRATION OF ENKEPHALIN IN RAT [J].
BELLUZZI, JD ;
GRANT, N ;
GARSKY, V ;
SARANTAKIS, D ;
WISE, CD ;
STEIN, L .
NATURE, 1976, 260 (5552) :625-626
[2]  
BELLUZZI JD, 1976, NEUR ABSTR, V2, P564
[3]   EVIDENCE FOR ANALGESIC ACTIVITY OF ENKEPHALIN IN MOUSE [J].
BUSCHER, HH ;
HILL, RC ;
ROMER, D ;
CARDINAUX, F ;
CLOSSE, A ;
HAUSER, D ;
PLESS, J .
NATURE, 1976, 261 (5559) :423-425
[4]   OPIATE RECEPTOR AFFINITIES AND BEHAVIORAL-EFFECTS OF ENKEPHALIN - STRUCTURE-ACTIVITY RELATIONSHIP OF 10 SYNTHETIC PEPTIDE ANALOGS [J].
CHANG, JK ;
FONG, BTW ;
PERT, A ;
PERT, CB .
LIFE SCIENCES, 1976, 18 (12) :1473-1481
[5]  
D'amour FE, 1941, J PHARMACOL EXP THER, V72, P74
[6]   ENCEPHALIN-INDUCED DEPRESSION OF SINGLE NEURONS IN BRAIN AREAS WITH OPIATE RECEPTORS-ANTAGONISM BY NALOXONE [J].
FREDERICKSON, RCA ;
NORRIS, FH .
SCIENCE, 1976, 194 (4263) :440-442
[7]   STEREOSPECIFIC AND NONSPECIFIC INTERACTIONS OF MORPHINE CONGENER LEVORPHANOL IN SUBCELLULAR FRACTIONS OF MOUSE BRAIN [J].
GOLDSTEIN, A ;
LOWNEY, LI ;
PAL, BK .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1971, 68 (08) :1742-+
[8]   MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].
HAMBROOK, JM ;
MORGAN, BA ;
RANCE, MJ ;
SMITH, CFC .
NATURE, 1976, 262 (5571) :782-783
[9]   IDENTIFICATION OF 2 RELATED PENTAPEPTIDES FROM BRAIN WITH POTENT OPIATE AGONIST ACTIVITY [J].
HUGHES, J ;
SMITH, TW ;
KOSTERLITZ, HW ;
FOTHERGILL, LA ;
MORGAN, BA ;
MORRIS, HR .
NATURE, 1975, 258 (5536) :577-579
[10]  
JACQUET YF, 1976, OPIATES ENDOGENOUS O