INTEGRATED QSAR OF H1-RECEPTOR ANTAGONISTS

被引:0
作者
REKKER, RF [1 ]
NAUTA, WT [1 ]
BULTSMA, T [1 ]
WARINGA, CG [1 ]
机构
[1] VRIJE UNIV AMSTERDAM,DEPT MED CHEM,DE BOELELAAN 1083,AMSTERDAM,NETHERLANDS
关键词
D O I
暂无
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:557 / 562
页数:6
相关论文
共 50 条
[41]   Role of histamine in the pathophysiology of asthma:: Immunomodulatory and antiinflammatory activities of H1-receptor antagonists [J].
Gelfaned, EW .
AMERICAN JOURNAL OF MEDICINE, 2002, 113 :2S-7S
[42]   PHARMACOLOGICAL CHARACTERIZATION OF CARDIAC HISTAMINE RECEPTORS - SENSITIVITY TO H1-RECEPTOR AND H2-RECEPTOR AGONISTS AND ANTAGONISTS [J].
LEVI, R ;
CAPURRO, N ;
LEE, CH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1975, 30 (02) :328-335
[43]   EFFECTS AND SIDE-EFFECTS OF H1-RECEPTOR AND H2-RECEPTOR ANTAGONISTS IN CLINICAL SITUATIONS - COMMENT [J].
SEWING, KF .
KLINISCHE WOCHENSCHRIFT, 1982, 60 (17) :1046-1047
[44]   CONGENITAL BULLOUS URTICARIA PIGMENTOSA - TREATMENT WITH CONCOMITANT USE OF H1-RECEPTOR AND H2-RECEPTOR ANTAGONISTS [J].
FENSKE, NA ;
LOBER, CW ;
PAUTLER, SE .
ARCHIVES OF DERMATOLOGY, 1985, 121 (01) :115-118
[45]   HISTAMINE-RELEASE WITH INTRAVENOUS NARCOTICS - PROTECTIVE EFFECTS OF H1-RECEPTOR AND H2-RECEPTOR ANTAGONISTS [J].
PHILBIN, DM ;
MOSS, J ;
ROSOW, CE ;
AKINS, CW ;
ROSENBERGER, JL .
KLINISCHE WOCHENSCHRIFT, 1982, 60 (17) :1056-1059
[46]   INHIBITION OF SYMPATHETIC NERVOUS-SYSTEM BY HISTAMINE - STUDIES WITH H1-RECEPTOR AND H2-RECEPTOR ANTAGONISTS [J].
LOKHANDWALA, MF .
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1978, 206 (01) :115-122
[47]   QSAR AND MOLECULAR MODELING STUDIES ON HISTAMINE H-1-RECEPTOR ANTAGONISTS [J].
TERLAAK, AM ;
VANDROOGE, MJ ;
TIMMERMAN, H ;
DENKELDER, GMD .
QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIPS, 1992, 11 (03) :348-363
[48]   Regulation of H1-receptor coupling and H1-receptor mRNA by histamine in bovine tracheal smooth muscle [J].
Pype, JL ;
Dupont, LJ ;
Mak, JCW ;
Barnes, PJ ;
Verleden, GM .
BRITISH JOURNAL OF PHARMACOLOGY, 1998, 123 (05) :984-990
[49]   CRYSTALLINE AND CONFORMATIONAL STUDIES ON HISTAMINE H1-RECEPTOR ANTAGONISTS .2. CYCLIZINE HYDROCHLORIDE [J].
BERTOLASI, V ;
BOREA, PA ;
GILLI, G ;
SACERDOTI, M .
ACTA CRYSTALLOGRAPHICA SECTION B-STRUCTURAL SCIENCE, 1980, 36 (AUG) :1975-1977