DYNAMICS OF A RECEPTOR-BOUND LIGAND BY HETERONUCLEAR NMR - FK506 BOUND TO FKBP-12

被引:17
作者
LEPRE, CA
CHENG, JW
MOORE, JM
机构
[1] Vertex Pharmaceuticals, Incorporated, Cambridge, Massachusetts 02139-4211
关键词
D O I
10.1021/ja00064a080
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:4929 / 4930
页数:2
相关论文
共 26 条
[1]  
ALDAPE RA, 1992, J BIOL CHEM, V267, P16029
[2]  
CHENG J, UNPUB
[3]   IDENTIFICATION OF CALCINEURIN AS A KEY SIGNALING ENZYME IN LYMPHOCYTE-T ACTIVATION [J].
CLIPSTONE, NA ;
CRABTREE, GR .
NATURE, 1992, 357 (6380) :695-697
[4]   CALCINEURIN PHOSPHATASE-ACTIVITY IN LYMPHOCYTES-T IS INHIBITED BY FK-506 AND CYCLOSPORINE-A [J].
FRUMAN, DA ;
KLEE, CB ;
BIERER, BE ;
BURAKOFF, SJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (09) :3686-3690
[5]  
KORDEL J, 1992, BIOCHEMISTRY-US, V31, P4856
[6]   SOLUTION STRUCTURE OF FK506 BOUND TO FKBP-12 [J].
LEPRE, CA ;
THOMSON, JA ;
MOORE, JM .
FEBS LETTERS, 1992, 302 (01) :89-96
[7]   MODEL-FREE APPROACH TO THE INTERPRETATION OF NUCLEAR MAGNETIC-RESONANCE RELAXATION IN MACROMOLECULES .2. ANALYSIS OF EXPERIMENTAL RESULTS [J].
LIPARI, G ;
SZABO, A .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1982, 104 (17) :4559-4570
[8]   MODEL-FREE APPROACH TO THE INTERPRETATION OF NUCLEAR MAGNETIC-RESONANCE RELAXATION IN MACROMOLECULES .1. THEORY AND RANGE OF VALIDITY [J].
LIPARI, G ;
SZABO, A .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1982, 104 (17) :4546-4559
[9]   CALCINEURIN IS A COMMON TARGET OF CYCLOPHILIN-CYCLOSPORINE-A AND FKBP-FK506 COMPLEXES [J].
LIU, J ;
FARMER, JD ;
LANE, WS ;
FRIEDMAN, J ;
WEISSMAN, I ;
SCHREIBER, SL .
CELL, 1991, 66 (04) :807-815
[10]   INHIBITION OF T-CELL SIGNALING BY IMMUNOPHILIN LIGAND COMPLEXES CORRELATES WITH LOSS OF CALCINEURIN PHOSPHATASE-ACTIVITY [J].
LIU, J ;
ALBERS, MW ;
WANDLESS, TJ ;
LUAN, S ;
ALBERG, DG ;
BELSHAW, PJ ;
COHEN, P ;
MACKINTOSH, C ;
KLEE, CB ;
SCHREIBER, SL .
BIOCHEMISTRY, 1992, 31 (16) :3896-3901