EFFECTS OF STEROID D-RING MODIFICATION ON SUICIDE INACTIVATION AND COMPETITIVE-INHIBITION OF AROMATASE BY ANALOGS OF ANDROSTA-1,4-DIENE-3,17-DIONE

被引：30

作者：

SHERWIN, PF ^{[1
]}

MCMULLAN, PC ^{[1
]}

COVEY, DF ^{[1
]}

机构：

[1] WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,ST LOUIS,MO 63110

来源：

关键词：

D O I：

10.1021/jm00123a026

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：651 / 658

页数：8

共 48 条

[1] SUICIDE ENZYME INACTIVATORS
ABELES, RH
[J]. CHEMICAL & ENGINEERING NEWS, 1983, 61 (38) : 48 - 56
[2] RESEARCHES ON ACETYLENIC COMPOUNDS .1. THE PREPARATION OF ACETYLENIC KETONES BY OXIDATION OF ACETYLENIC CARBINOLS AND GLYCOLS
BOWDEN, K
HEILBRON, IM
JONES, ERH
WEEDON, BCL
[J]. JOURNAL OF THE CHEMICAL SOCIETY, 1946, (JAN): : 39 - 45
[3] BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[4] COREY EJ, 1975, TETRAHEDRON LETT, P2647
[5] COVEY DF, 1982, CANCER RES, V42, P3327
[6] COVEY DF, 1981, J BIOL CHEM, V256, P1076
[7] COVEY DF, 1988, STEROID BIOSYNTHESIS, P534
[8] DEMONTELLANO PRO, 1986, CYTOCHROME P450 STRU, P273
[9] DISALLE E, 1987, Patent No. 3622841
[10] THE BROMINATION OF 3-KETOSTEROIDS IN ACETIC ACID AND THE EFFECT OF TRACE SUBSTANCES IN THE SOLVENT
DJERASSI, C
SCHOLZ, CR
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1947, 69 (10) : 2404 - 2410