CHARACTERIZATION OF THE CARDIOVASCULAR EFFECTS OF R-ALPHA-METHYL HISTAMINE, A SELECTIVE HISTAMINE-H-3 RECEPTOR AGONIST, IN ANESTHETIZED RATS

被引:0
|
作者
HEGDE, SS [1 ]
CHAN, P [1 ]
EGLEN, RM [1 ]
机构
[1] SYNTEX INC,DISCOVERY RES,PALO ALTO,CA 94304
来源
FASEB JOURNAL | 1993年 / 7卷 / 04期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:A620 / A620
页数:1
相关论文
共 50 条
  • [31] ANALEPTIC EFFECT OF CENTRALLY ADMINISTERED HISTAMINE H2-RECEPTOR AGONIST DIMAPRIT BUT NOT IMPROMIDINE IN URETHANE-ANESTHETIZED RATS
    PAAKKARI, I
    KARPPANEN, H
    NEUROPHARMACOLOGY, 1982, 21 (02) : 171 - 178
  • [32] Enzyme-catalyzed prodrug approaches for the histamine H3-receptor agonist (R)-α-methylhistamine
    Stark, H
    Krause, M
    Rouleau, A
    Garbarg, M
    Schwartz, JC
    Schunack, W
    BIOORGANIC & MEDICINAL CHEMISTRY, 2001, 9 (01) : 191 - 198
  • [33] Acute central administration of immepip, a histamine H3 receptor agonist, suppresses hypothalamic histamine release and elicits feeding behavior in rats
    Chiba, Seiichi
    Itateyama, Emi
    Sakata, Toshiie
    Yoshimatsu, Hironobu
    BRAIN RESEARCH BULLETIN, 2009, 79 (01) : 37 - 40
  • [34] EFFECTS OF SELECTIVE ACTIVATION OR BLOCKADE OF THE HISTAMINE-H3 RECEPTOR ON SLEEP AND WAKEFULNESS
    MONTI, JM
    JANTOS, H
    BOUSSARD, M
    ALTIER, H
    ORELLANA, C
    OLIVERA, S
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 205 (03) : 283 - 287
  • [35] Molecular Determinants of Selective Agonist and Antagonist Binding to the Histamine H4 Receptor
    Istyastono, Enade P.
    de Graaf, Chris
    de Esch, Iwan J. P.
    Leurs, Rob
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2011, 11 (06) : 661 - 679
  • [36] CHARACTERIZATION OF THE HIGH-AFFINITY BINDING-SITES OF [HISTAMINE-H-3 IN RAT-BRAIN
    BARBIN, G
    PALACIOS, JM
    RODERGAS, E
    SCHWARTZ, JC
    GARBARG, M
    MOLECULAR PHARMACOLOGY, 1980, 18 (01) : 1 - 10
  • [37] EFFECTS OF N-ALPHA-METHYL HISTAMINE ON THE ISOLATED GUINEA-PIG HEART, EVIDENCE FOR H3-HISTAMINE RECEPTORS
    ANDJELKOVIC, IZ
    COLLIS, CS
    ROSIC, MA
    SEGAL, MB
    ZLOKOVIC, BZ
    JOURNAL OF PHYSIOLOGY-LONDON, 1990, 424 : P58 - P58
  • [38] Highlights in cardiovascular effects of histamine and H-1-receptor antagonists
    Genovese, A
    Spadaro, G
    ALLERGY, 1997, 52 : 67 - 78
  • [39] Effects of histamine H1R-H4R-agonist on the airway epithelium of rabbits
    Dilkash, Naushad A.
    Tripathi, Trivendra
    Khan, Aijaz Ahmed
    Shahid, Mohd
    Khan, Haris M.
    Siddiqui, Mashiatullah
    Khan, Rahat Ali
    ASIAN PACIFIC JOURNAL OF TROPICAL MEDICINE, 2010, 3 (05) : 367 - 370
  • [40] CARDIAC EFFECTS OF AMTHAMINE - A NEW HISTAMINE H-2-RECEPTOR AGONIST
    CORUZZI, G
    GAMBARELLI, E
    TIMMERMAN, H
    EUROPEAN JOURNAL OF CLINICAL INVESTIGATION, 1995, 25 : 27 - 28