CHARACTERIZATION OF THE CARDIOVASCULAR EFFECTS OF R-ALPHA-METHYL HISTAMINE, A SELECTIVE HISTAMINE-H-3 RECEPTOR AGONIST, IN ANESTHETIZED RATS

被引:0
|
作者
HEGDE, SS [1 ]
CHAN, P [1 ]
EGLEN, RM [1 ]
机构
[1] SYNTEX INC,DISCOVERY RES,PALO ALTO,CA 94304
来源
FASEB JOURNAL | 1993年 / 7卷 / 04期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:A620 / A620
页数:1
相关论文
共 50 条
  • [11] BINDING OF [HISTAMINE-H-3 TO RECEPTOR-SITES IN RAT-BRAIN
    SINGH, VK
    MCGEER, EG
    EXPERIMENTAL NEUROLOGY, 1979, 66 (02) : 413 - 418
  • [12] EFFECTS OF DIFFERENT TYPES OF STRESS ON HISTAMINE-H-3, RECEPTORS IN THE RAT CORTEX
    GHI, P
    CARLO, FB
    BLENGIO, M
    BRAIN RESEARCH, 1995, 690 (01) : 104 - 107
  • [13] DIMAPRIT, A SELECTIVE HISTAMINE-H2-RECEPTOR AGONIST, REDUCES PROLACTIN LEVELS IN RATS
    FALASCHI, P
    DURSO, R
    FRAJESE, G
    RUGGIERI, S
    SCARNATI, E
    FORCHETTI, C
    AGNOLI, A
    ACTA ENDOCRINOLOGICA, 1979, 91 : 161 - 161
  • [14] Discovery and characterization of CEP-26401: A potent, selective histamine H3 receptor inverse agonist
    Hudkins, Robert L.
    Raddatz, Rita
    Tao, Ming
    Mathiasen, Joanne R.
    Grunner, John A.
    Aimone, Lisa D.
    Prouty, Catherine P.
    Becknell, Nadine C.
    Knutsen, Lars
    Yazdanian, Mehran
    Moachon, Gilbert
    Ator, Mark A.
    Mallamo, John P.
    Marino, Michael J.
    Bacon, Edward R.
    Williams, Michael
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241
  • [15] AMSELAMINE, A NEW SELECTIVE HISTAMINE H-2-RECEPTOR AGONIST
    VANDERGOOT, H
    ERIKS, JC
    LEURS, R
    TIMMERMAN, H
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1994, 4 (16) : 1913 - 1916
  • [16] INHIBITORY EFFECTS OF HISTAMINE H3 RECEPTOR (H3R) INVERSE AGONIST/ANTAGONIST ON MICROGLIAL FUNCTIONS
    Iida, T.
    Yoshikawa, T.
    Yanai, K.
    INFLAMMATION RESEARCH, 2018, 67 : S25 - S25
  • [17] EFFECTS OF THE HISTAMINE H3-AGONIST (R)-ALPHA-METHYLHISTAMINE AND THE ANTAGONIST THIOPERAMIDE ON HISTAMINE-METABOLISM IN THE MOUSE AND RAT-BRAIN
    OISHI, R
    ITOH, Y
    NISHIBORI, M
    SAEKI, K
    JOURNAL OF NEUROCHEMISTRY, 1989, 52 (05) : 1388 - 1392
  • [18] THE SELECTIVE HISTAMINE H-1-RECEPTOR AGONIST 2-(3-TRIFLUOROMETHYLPHENYL)HISTAMINE INCREASES WAKING IN THE RAT
    MONTI, JM
    JANTOS, H
    LESCHKE, C
    ELZ, S
    SCHUNACK, W
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 1994, 4 (04) : 459 - 462
  • [19] CARDIOVASCULAR EFFECTS IN MAN OF IMPROMIDINE, A NOVEL AND SPECIFIC HISTAMINE H-2-RECEPTOR AGONIST
    BOYCE, MJ
    BALASUBRAMANIAN, V
    WAREHAM, K
    BRITISH JOURNAL OF PHARMACOLOGY, 1980, 70 (01) : P157 - P158
  • [20] Effects of histamine H3 receptor agonist and antagonist on histamine co-transmitter expression in rat brain
    C. Chotard
    T. Ouimet
    S. Morisset
    U. Sahm
    J. C. Schwartz
    S. Trottier
    Journal of Neural Transmission, 2002, 109 : 293 - 306