RECEPTOR-BINDING AND BIOLOGICAL-ACTIVITY OF STEROIDAL AND NON-STEROIDAL ANTIANDROGENS

被引：84
作者：
WAKELING, AE
FURR, BJA
GLEN, AT
HUGHES, LR
机构：
来源：
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY | 1981年 / 15卷 / DEC期
关键词：
D O I：
10.1016/0022-4731(81)90297-1
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：355 / 359
页数：5
相关论文
共 16 条
[1]   ASSAY OF ANDROGEN BINDING-SITES BY EXCHANGE WITH METHYLTRIENOLONE (R 1881) [J].
BONNE, C ;
RAYNAUD, JP .
STEROIDS, 1976, 27 (04) :497-507
[2]   METHYLTRIENOLONE, A SPECIFIC LIGAND FOR CELLULAR ANDROGEN RECEPTORS [J].
BONNE, C ;
RAYNAUD, JP .
STEROIDS, 1975, 26 (02) :227-232
[3]   HIGH-AFFINITY BINDING TO THE ESTROGEN-RECEPTOR OF [4-HYDROXYTAMOXIFEN-H-3, AN ACTIVE ANTI-ESTROGEN METABOLITE [J].
BORGNA, JL ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1980, 20 (01) :71-85
[4]   COMPARATIVE-STUDY OF ANTIESTROGEN ACTION - TEMPORAL PATTERNS OF ANTAGONISM OF ESTROGEN STIMULATED UTERINE GROWTH AND EFFECTS ON ESTROGEN-RECEPTOR LEVELS [J].
FERGUSON, ER ;
KATZENELLENBOGEN, BS .
ENDOCRINOLOGY, 1977, 100 (05) :1242-1251
[5]  
Furr BJ, 1979, PHARMACOLOGICAL BIOC, V2, P355
[6]   DISPOSITION OF A NEW, NONSTEROID, ANTIANDROGEN, ALPHA,ALPHA,ALPHA-TRIFLUORO-2-METHYL-4'-NITRO-M-PROPIONOTOLUIDIDE (FLUTAMIDE), IN MEN FOLLOWING A SINGLE ORAL 200 MG DOSE [J].
KATCHEN, B ;
BUXBAUM, S .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1975, 41 (02) :373-379
[7]   ACTION OF A NONSTEROIDAL ANTIANDROGEN, FLUTAMIDE, ON RECEPTOR-BINDING AND NUCLEAR RETENTION OF 5-ALPHA DIHYDROTESTOSTERONE IN RAT VENTRAL PROSTATE [J].
LIAO, S ;
HOWELL, DK ;
CHANG, TM .
ENDOCRINOLOGY, 1974, 94 (04) :1205-1209
[8]   Anti-Androgenicity of Flutamide and its Metabolite Sch 16423 [J].
Neri, Rudolph ;
Peets, Edwin ;
Watnick, Arthur .
BIOCHEMICAL SOCIETY TRANSACTIONS, 1979, 7 :565-569
[9]  
Neumann F, 1977, ANDROGENS ANTIANDROG, P163
[10]   CONCENTRATIONS OF PUTRESCINE AND POLYAMINES AND THEIR ENZYMIC SYNTHESIS DURING ANDROGEN-INDUCED PROSTATIC GROWTH [J].
PEGG, AE ;
LOCKWOOD, DH ;
WILLIAMS.HG .
BIOCHEMICAL JOURNAL, 1970, 117 (01) :17-&
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