CORRELATION OF THE HYPNOTIC POTENCY OF BENZODIAZEPINES WITH INHIBITION OF VOLTAGE-DEPENDENT CALCIUM-UPTAKE INTO MOUSE-BRAIN SYNAPTOSOMES

被引:19
作者
LESLIE, SW [1 ]
CHANDLER, LJ [1 ]
CHWEH, AY [1 ]
SWINYARD, EA [1 ]
机构
[1] UNIV UTAH,COLL PHARM,DEPT BIOCHEM PHARMACOL & TOXICOL,SALT LAKE CITY,UT 84112
关键词
D O I
10.1016/0014-2999(86)90748-X
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:129 / 134
页数:6
相关论文
共 24 条
[1]   CA-2+-ANTAGONISTIC EFFECTS OF FLURAZEPAM, A BENZODIAZEPINE DERIVATIVE, ON ISOLATED GUINEA-PIG LEFT ATRIA [J].
AKUTAGAWA, K ;
MAKINO, M ;
ISHII, K .
JAPANESE JOURNAL OF PHARMACOLOGY, 1983, 33 (04) :845-850
[2]   GABA AGONISTS AND ANTAGONISTS [J].
ANDREWS, PR ;
JOHNSTON, GAR .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (18) :2697-2702
[3]   EFFECT OF GABA AGONISTS ON THE NEUROTOXICITY AND ANTICONVULSANT ACTIVITY OF BENZODIAZEPINES [J].
CHWEH, AY ;
SWINYARD, EA ;
WOLF, HH ;
KUPFERBERG, HJ .
LIFE SCIENCES, 1985, 36 (08) :737-744
[4]   CORRELATIONS AMONG MINIMAL NEUROTOXICITY, ANTI-CONVULSANT ACTIVITY, AND DISPLACING POTENCIES IN [FLUNITRAZEPAM-H-3 BINDING OF BENZODIAZEPINES [J].
CHWEH, AY ;
SWINYARD, EA ;
WOLF, HH ;
KUPFERBERG, HJ .
EPILEPSIA, 1983, 24 (06) :668-677
[5]   HYPNOTIC ACTION OF BENZODIAZEPINES - A POSSIBLE MECHANISM [J].
CHWEH, AY ;
LIN, YB ;
SWINYARD, EA .
LIFE SCIENCES, 1984, 34 (18) :1763-1768
[6]   MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 :531-545
[7]  
Cotman C W, 1974, Methods Enzymol, V31, P445
[8]   BENZODIAZEPINE INHIBITION OF THE CALCIUM-CALMODULIN PROTEIN-KINASE SYSTEM IN BRAIN MEMBRANE [J].
DELORENZO, RJ ;
BURDETTE, S ;
HOLDERNESS, J .
SCIENCE, 1981, 213 (4507) :546-549
[9]   THE CALMODULIN HYPOTHESIS OF NEUROTRANSMISSION [J].
DELORENZO, RJ .
CELL CALCIUM, 1981, 2 (04) :365-385
[10]  
ELROD SV, 1980, J PHARMACOL EXP THER, V212, P131