SYNTHESIS AND CHARACTERIZATION OF IODINATED VASOPRESSIN ANTAGONISTS WHICH RETAIN HIGH-AFFINITY FOR THE VASOPRESSIN RECEPTOR

被引：16

作者：

MOORE, ML

HUFFMAN, WF

ROBERTS, GD

ROTTSCHAEFER, S

SULAT, L

STEFANKIEWICZ, JS

STASSEN, F

机构：

来源：

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS | 1984年 / 121卷 / 03期

关键词：

D O I：

10.1016/0006-291X(84)90759-9

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：878 / 883

页数：6

共 7 条

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[2] [1-(BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENEPROPIONIC ACID),2-(O-METHYL)TYROSINE]ARGININE-VASOPRESSIN AND [1-(BETA-MERCAPTO-BETA,BETA-CYCLOPENTAMETHYLENEPROPIONIC ACID)]ARGININE-VASOPRESSIN, 2 HIGHLY POTENT ANTAGONISTS OF THE VASOPRESSOR RESPONSE TO ARGININE-VASOPRESSIN [J].

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LAMMEK, B ;

MANNING, M ;

SETO, J ;

HALDAR, J ;

SAWYER, WH .

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[3] DESIGN OF MORE POTENT AND SELECTIVE ANTAGONISTS OF THE ANTI-DIURETIC RESPONSES TO ARGININE-VASOPRESSIN DEVOID OF ANTI-DIURETIC AGONISM [J].

MANNING, M ;

KLIS, WA ;

OLMA, A ;

SETO, J ;

SAWYER, WH .

JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (04) :414-419

[4]

MATTERA R, 1982, INT J PEPT PROT RES, V19, P172

[5]

STASSEN FL, 1982, J PHARMACOL EXP THER, V223, P50

[6]

VANBRUSSEL Y, 1983, J LABELLED COMP RADI, V20, P89

[7] CHEMISTRY AND STRUCUTRE-ACTIVITY RELATIONS OF ANTIDIURETIC HORMONES [J].

WALTER, R ;

RUDINGER, J ;

SCHWARTZ, IL .

AMERICAN JOURNAL OF MEDICINE, 1967, 42 (05) :653-+

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