SYNTHESIS AND ANTI-HIV ACTIVITY OF VARIOUS 2'-SUBSTITUTED AND 3'-SUBSTITUTED 2',3'-DIDEOXYADENOSINES - A STRUCTURE ACTIVITY ANALYSIS

被引：177

作者：

HERDEWIJN, P ^{[1
]}

PAUWELS, R ^{[1
]}

BABA, M ^{[1
]}

BALZARINI, J ^{[1
]}

DECLERCQ, E ^{[1
]}

机构：

[1] CATHOLIC UNIV LEUVEN, REGA INST MED RES, B-3000 LOUVAIN, BELGIUM

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1987年 / 30卷 / 11期

关键词：

D O I：

10.1021/jm00394a034

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2131 / 2137

页数：7

共 31 条

[1] INHIBITION BY 2',3'-DIDEOXYTHYMIDINE OF RETROVIRAL INFECTION OF MOUSE AND HUMAN-CELLS
FURMANSKI, P
BOURGUIGNON, GJ
BOLLES, CS
COROMBOS, JD
DAS, MR
[J]. CANCER LETTERS, 1980, 8 (04) : 307 - 315
[2] NITRATE ION AS CATALYST FOR SELECTIVE SILYLATIONS OF NUCLEOSIDES
HAKIMELAHI, GH
PROBA, ZA
OGILVIE, KK
[J]. TETRAHEDRON LETTERS, 1981, 22 (48) : 4775 - 4778
[3] NUCLEIC-ACID RELATED-COMPOUNDS .49. REGIOSPECIFIC AND STEREOSELECTIVE CONVERSION OF RIBONUCLEOSIDES TO 3'-DEOXYNUCLEOSIDES - A HIGH-YIELD 3-STAGE SYNTHESIS OF CORDYCEPIN FROM ADENOSINE
HANSSKE, F
ROBINS, MJ
[J]. TETRAHEDRON LETTERS, 1985, 26 (36) : 4295 - 4298
[4] NUCLEIC-ACID RELATED-COMPOUNDS .45. A DEOXYGENATIVE [1,2]-HYDRIDE SHIFT REARRANGEMENT CONVERTING CYCLIC CIS-DIOL MONOTOSYLATES TO INVERTED SECONDARY ALCOHOLS
HANSSKE, F
ROBINS, MJ
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1983, 105 (22) : 6736 - 6737
[5] 3'-SUBSTITUTED 2',3'-DIDEOXYNUCLEOSIDE ANALOGS AS POTENTIAL ANTI-HIV (HTLV-III/LAV) AGENTS
HERDEWIJN, P
BALZARINI, J
DECLERCQ, E
PAUWELS, R
BABA, M
BRODER, S
VANDERHAEGHE, H
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (08) : 1270 - 1278
[6] IKEHARA M, 1978, CHEM PHARM BULL, V26, P2449
[7] SYNTHESIS OF 3'-AZIDO-2',3'-DIDEOXYRIBOFURANOSYLPURINES
IMAZAWA, M
ECKSTEIN, F
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1978, 43 (15) : 3044 - 3048
[8] KLECKER RW, IN PRESS CLIN PHARM
[9] INVOLVEMENT OF EUKARYOTIC DEOXYRIBONUCLEIC-ACID POLYMERASE-ALPHA AND POLYMERASE-GAMMA IN THE REPLICATION OF CELLULAR AND VIRAL DEOXYRIBONUCLEIC-ACID
KROKAN, H
SCHAFFER, P
DEPAMPHILIS, ML
[J]. BIOCHEMISTRY, 1979, 18 (20) : 4431 - 4443
[10] Langen P, 1969, Acta Biol Med Ger, V23, P759

← 1 2 3 4 →