NOVEL, NONPEPTIDAL GASTRIN/CCK-B RECEPTOR ANTAGONISTS

被引：0
|
作者：
FREIDINGER, RM [1 ]
BOCK, MB [1 ]
DIPARDO, RM [1 ]
EVANS, BE [1 ]
RITTLE, KE [1 ]
VEBER, DF [1 ]
CHANG, RSL [1 ]
LOTTI, VJ [1 ]
机构：
[1] MERCK SHARP & DOHME RES LABS,W POINT,PA 19486
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 1988年 / 195卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：5 / BIOL
相关论文
共 50 条
  • [21] Immunohistochemical localization of the gastrin/CCK-B receptor in the rat stomach
    Song, M
    Wong, H
    Ohning, G
    Walsh, JH
    GASTROENTEROLOGY, 1996, 110 (04) : A1120 - A1120
  • [22] Nuclear expression of an epitope of the CCK-B/gastrin receptor.
    Caplin, ME
    Khan, K
    Michaeli, D
    Lewin, J
    Savage, K
    Watson, SA
    Pounder, RE
    Dhillon, AP
    GASTROENTEROLOGY, 1997, 112 (04) : A1136 - A1136
  • [23] CHOLECYSTOKININ DIPEPTOID ANTAGONISTS - DESIGN, SYNTHESIS, AND ANXIOLYTIC PROFILE OF SOME NOVEL CCK-A AND CCK-B SELECTIVE AND MIXED CCK-A CCK-B ANTAGONISTS
    BODEN, PR
    HIGGINBOTTOM, M
    HILL, DR
    HORWELL, DC
    HUGHES, J
    REES, DC
    ROBERTS, E
    SINGH, L
    SUMANCHAUHAN, N
    WOODRUFF, GN
    JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (05) : 552 - 565
  • [24] SYNTHESIS AND SAR STUDY OF NOVEL CCK-B ANTAGONISTS
    PADIA, JK
    BOLTON, GL
    HILL, D
    HORWELL, DC
    ROTH, BD
    TRIVEDI, BK
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1993, 3 (12) : 2805 - 2810
  • [25] SYNTHESIS AND SAR STUDY OF NOVEL CCK-B ANTAGONISTS
    PADIA, JK
    BOLTON, GL
    HILL, D
    HORWELL, DC
    ROTH, BD
    TRIVEDI, BK
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1992, 204 : 90 - MEDI
  • [26] CCK-B/GASTRIN RECEPTOR MEDIATES GASTRIN, CCK BUT NOT HISTAMINE STIMULATING ACID-SECRETION IN RATS
    SONG, Y
    LI, P
    LEE, KY
    CHEY, WY
    GASTROENTEROLOGY, 1994, 106 (04) : A843 - A843
  • [27] Novel nonpeptide CCK-B antagonists: Design and development of quinazolinone derivatives as potent, selective, and orally active CCK-B antagonists
    Padia, JK
    Field, M
    Hinton, J
    Meecham, K
    Pablo, J
    Pinnock, R
    Roth, BD
    Singh, L
    Suman-Chauhan, N
    Trivedi, BK
    Webdale, L
    JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (07) : 1042 - 1049
  • [28] CLASS-SPECIFIC DIFFERENCES IN RECEPTOR-BINDING AND GASTRIC ANTISECRETORY ACTIVITY OF GASTRIN CCK-B RECEPTOR ANTAGONISTS
    PENDLEY, C
    EWING, W
    MOLINO, B
    GUYON, C
    DUBROEUCQ, MC
    MARTIN, G
    FASEB JOURNAL, 1993, 7 (03): : A23 - A23
  • [29] Characterization of the CCK-B/gastrin receptor on human gastric cancer cells
    Shih, AH
    Wotring, MG
    Smith, MP
    Zagon, IS
    Smith, JP
    GASTROENTEROLOGY, 1996, 110 (04) : A1118 - A1118
  • [30] CENTRALLY ADMINISTERED CCK PRODUCES ANTINOCICEPTION THAT IS NOT BLOCKED BY CCK-A OR CCK-B RECEPTOR ANTAGONISTS
    WILLIAMS, CL
    ROSENFELD, GC
    BURKS, TF
    FASEB JOURNAL, 1994, 8 (05): : A627 - A627
12345