Synthesis of a new pyrrolo[1,3]diazepine: 4H-pyrrolo[1,2-a]thieno[2,3-e][1,3]diazepine

被引：4

作者：

Daich, A

Ohier, P

Decroix, B

机构：

[1] Laboratoire de Chimie, Faculté des Sciences et des Techniques, Université du Havre, Le Havre, 76600

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1995年 / 32卷 / 06期

关键词：

D O I：

10.1002/jhet.5570320611

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The 4H-pyrrolo[1,2-a]thieno[2,3-e][1,3]diazepine (20) was synthesized by the one-pot intramolecular cyclization of the appropriate nitroaldehyde 13. This key intermediate 13 was obtained by two pathways from methyl 3-bromomethylthiophene-2-carboxylate (6).

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页码：1731 / 1734

页数：4

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