USE OF [H-3] TRIMETOQUINOL AS A RADIOLIGAND IN HUMAN-PLATELETS - INTERACTION WITH PUTATIVE ENDOPEROXIDE THROMBOXANE-A2 RECEPTOR-SITES

被引:10
作者
AHN, CH
WALLACE, LJ
MILLER, DD
FELLER, DR
机构
[1] OHIO STATE UNIV,COLL PHARM,DIV MED CHEM,COLUMBUS,OH 43210
[2] OHIO STATE UNIV,COLL PHARM,DIV PHARMACOL,COLUMBUS,OH 43210
关键词
D O I
10.1016/0049-3848(88)90268-X
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:387 / 399
页数:13
相关论文
共 24 条
[1]  
AHN CH, 1985, THESIS OHIO STATE U
[2]   LIGAND-BINDING TO THROMBOXANE RECEPTORS ON HUMAN-PLATELETS - CORRELATION WITH BIOLOGICAL-ACTIVITY [J].
ARMSTRONG, RA ;
JONES, RL ;
WILSON, NH .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 79 (04) :953-964
[3]   AGGREGATION OF BLOOD PLATELETS BY ADENOSINE DIPHOSPHATE AND ITS REVERSAL [J].
BORN, GVR .
NATURE, 1962, 194 (4832) :927-&
[4]   COMPARISON OF THE ACTIONS OF U-46619, A PROSTAGLANDIN H2-ANALOGUE, WITH THOSE OF PROSTAGLANDIN-H2 AND THROMBOXANE-A2 ON SOME ISOLATED SMOOTH-MUSCLE PREPARATIONS [J].
COLEMAN, RA ;
HUMPHREY, PPA ;
KENNEDY, I ;
LEVY, GP ;
LUMLEY, P .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 73 (03) :773-778
[5]   TRIMETHOQUINOL - DIFFERENT PHARMACOLOGICAL PROPERTIES OF OPTICAL ISOMERS [J].
DALTON, C ;
CROWLEY, HJ ;
CZYZEWSKI, LB .
BIOCHEMICAL PHARMACOLOGY, 1976, 25 (19) :2209-2210
[6]   A NOVEL-APPROACH FOR THE STUDY OF THROMBOXANE-A2 AND PROSTAGLANDIN-H2 RECEPTORS USING AN I-125-LABELED LIGAND [J].
HALUSHKA, PV ;
MACDERMOT, J ;
KNAPP, DR ;
ELLER, T ;
SAUSSY, DL ;
MAIS, D ;
BLAIR, IA ;
DOLLERY, CT .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (08) :1165-1170
[7]  
HALUSHKA PV, 1987, FASEB J, V46, P149
[8]   PROSTAGLANDIN ENDOPEROXIDES - NOVEL TRANSFORMATIONS OF ARACHIDONIC-ACID IN HUMAN PLATELETS [J].
HAMBERG, M ;
SAMUELSS.B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1974, 71 (09) :3400-3404
[9]   THROMBOXANES - NEW GROUP OF BIOLOGICALLY-ACTIVE COMPOUNDS DERIVED FROM PROSTAGLANDIN ENDOPEROXIDES [J].
HAMBERG, M ;
SVENSSON, J ;
SAMUELSSON, B .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1975, 72 (08) :2994-2998
[10]  
Harrold M W, 1987, Drug Des Deliv, V1, P193