A UNIQUELY POTENT RENIN INHIBITOR AND ITS UNANTICIPATED PLASMA-BINDING COMPONENT

被引：15

作者：

EVANS, BE ^{[1
]}

RITTLE, KE ^{[1
]}

BOCK, MG ^{[1
]}

BENNETT, CD ^{[1
]}

DIPARDO, RM ^{[1
]}

BOGER, J ^{[1
]}

POE, M ^{[1
]}

ULM, EH ^{[1
]}

LAMONT, BI ^{[1
]}

BLAINE, EH ^{[1
]}

FANELLI, GM ^{[1
]}

STABILITO, II ^{[1
]}

VEBER, DF ^{[1
]}

机构：

[1] MERCK SHARP & DOHME RES LABS,RAHWAY,NJ 07065

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1985年 / 28卷 / 12期

关键词：

D O I：

10.1021/jm00150a001

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1755 / 1756

页数：2

共 17 条

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[3]

BOGER J, 1983, PEPTIDES STRUCTURE F, P569

[4] COMPETITIVE INHIBITORS OF RENIN INHIBITORS EFFECTIVE AT PHYSIOLOGICAL PH [J].

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[5] A SUBSTRATE-ANALOG INHIBITOR OF RENIN THAT IS EFFECTIVE INVIVO [J].

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[6] SOLUBLE PEPSTATINS - NEW APPROACH TO BLOCKADE INVIVO OF THE RENIN-ANGIOTENSIN SYSTEM [J].

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[7]

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[8] COMPETITIVE INHIBITORS OF RENIN [J].

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BIOCHEMISTRY, 1973, 12 (20) :3877-3882

[9] SPECIFICITY OF HUMAN RENIN - STUDIES WITH PEPTIDE INHIBITORS [J].

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[10] SYNTHESIS OF ANALOGS OF THE CARBOXYL PROTEASE INHIBITOR PEPSTATIN - EFFECT OF STRUCTURE ON INHIBITION OF PEPSIN AND RENIN [J].

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