INTERACTION OF SPIRONOLACTONE AND DIGITALIS WITH 5ALPHA-DIHYDROTESTOSTERONE (DHT) 17 "BETA-HYDROXY-5ALPHA-ANDROSTAN-3-ONE (5ALPHA-DIHYDROTESTOSTERONE,DHT) RECEPTOR OF RAT VENTRAL PROSTATE

被引:67
作者
PITA, JC
LIPPMAN, ME
THOMPSON, EB
LORIAUX, DL
机构
[1] NCI,MED BRANCH,BETHESDA,MD 20014
[2] NCI,LAB BIOCHEM,BETHESDA,MD 20014
[3] NICHHD,REPRODUCTION BRANCH,BETHESDA,MD 20014
关键词
D O I
10.1210/endo-97-6-1521
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:1521 / 1527
页数:7
相关论文
共 35 条
[1]  
ANDERSON KM, 1968, NATURE, V196, P36
[2]   ANTIANDROGENIC EFFECT OF SPIRONOLACTONE IN RATS [J].
BASINGER, GT ;
GITTES, RF .
JOURNAL OF UROLOGY, 1974, 111 (01) :77-80
[3]   A PROSTATIC CYTOSOL RECEPTOR [J].
BAULIEU, EE ;
JUNG, I .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1970, 38 (04) :599-&
[4]   MODE OF SPIRONOLACTONE ANTI-ANDROGENIC ACTION - INHIBITION OF ANDROSTANOLONE BINDING TO RAT PROSTATE ANDROGEN RECEPTOR [J].
BONNE, C ;
RAYNAUD, JP .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1974, 2 (01) :59-67
[5]  
BRICKHARDT D, 1968, ANN INT MED, V68, P1069
[6]  
CASTLE MC, 1973, DRUG METAB DISPOS, V1, P590
[7]   DOUBLE-BLIND, CONTROLLED, CLINICAL TRIAL OF SPIRONOLACTONE FOR BENIGN PROSTATIC HYPERTROPHY [J].
CASTRO, JE ;
GRIFFITHS, HJ ;
EDWARDS, DE .
BRITISH JOURNAL OF SURGERY, 1971, 58 (07) :485-+
[8]   PROTAMINE-PRECIPITATED ESTROGEN-RECEPTOR - SOLID-PHASE LIGAND-EXCHANGE ASSAY [J].
CHAMNESS, GC ;
HUFF, K ;
MCGUIRE, WL .
STEROIDS, 1975, 25 (05) :627-635
[9]  
CLARCK E, 1965, JAMA-J AM MED ASSOC, V193, P157
[10]  
DOHERTY JE, 1973, ANN INTERN MED, V79, P229, DOI 10.7326/0003-4819-79-2-229