ANTINOCICEPTIVE POTENCIES OF BETA-CASOMORPHIN ANALOGS AS COMPARED TO THEIR AFFINITIES TOWARDS MU- AND DELTA- OPIATE RECEPTOR-SITES IN BRAIN AND PERIPHERY

被引：96
作者：
BRANTL, V
PFEIFFER, A
HERZ, A
HENSCHEN, A
LOTTSPEICH, F
机构：
[1] MAX PLANCK INST PSYCHIAT,DEPT NEUROPHARMACOL,D-8000 MUNICH 40,FED REP GER
[2] MAX PLANCK INST BIOCHEM,D-8033 MARTINSRIED,FED REP GER
来源：
PEPTIDES | 1982年 / 3卷 / 05期
关键词：
D O I：
10.1016/0196-9781(82)90017-1
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：793 / 797
页数：5
相关论文
共 26 条
[1]   MATERIAL WITH OPIOID ACTIVITY IN BOVINE-MILK AND MILK-PRODUCTS [J].
BRANTL, V ;
TESCHEMACHER, H .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 306 (03) :301-304
[2]   NOVEL OPIOID PEPTIDES DERIVED FROM CASEIN (BETA-CASOMORPHINS) .1. ISOLATION FROM BOVINE CASEIN PEPTONE [J].
BRANTL, V ;
TESCHEMACHER, H ;
HENSCHEN, A ;
LOTTSPEICH, F .
HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1979, 360 (09) :1211-1216
[3]   OPIOID ACTIVITIES OF BETA-CASOMORPHINS [J].
BRANTL, V ;
TESCHEMACHER, H ;
BLASIG, J ;
HENSCHEN, A ;
LOTTSPEICH, F .
LIFE SCIENCES, 1981, 28 (17) :1903-1909
[4]  
CHANG KJ, 1979, J BIOL CHEM, V254, P2610
[5]   MORPHICEPTIN (NH4-TYR-PRO-PHE-PRO-CONH2) - A POTENT AND SPECIFIC AGONIST FOR MORPHINE (MU) RECEPTORS [J].
CHANG, KJ ;
KILLIAN, A ;
HAZUM, E ;
CUATRECASAS, P ;
CHANG, JK .
SCIENCE, 1981, 212 (4490) :75-77
[6]   NOVEL OPIATE BINDING-SITES SELECTIVE FOR BENZOMORPHAN DRUGS [J].
CHANG, KJ ;
HAZUM, E ;
CUATRECASAS, P .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (07) :4141-4145
[7]   METKEPHAMID, A SYSTEMICALLY ACTIVE ANALOG OF METHIONINE ENKEPHALIN WITH POTENT OPIOID DELTA-RECEPTOR ACTIVITY [J].
FREDERICKSON, RCA ;
SMITHWICK, EL ;
SHUMAN, R ;
BEMIS, KG .
SCIENCE, 1981, 211 (4482) :603-605
[8]   EVIDENCE OF THE PREFERENTIAL INVOLVEMENT OF MU-RECEPTORS IN ANALGESIA USING ENKEPHALINS HIGHLY SELECTIVE FOR PERIPHERAL MU-RECEPTOR OR DELTA-RECEPTOR [J].
GACEL, G ;
FOURNIEZALUSKI, MC ;
FELLION, E ;
ROQUES, BP .
JOURNAL OF MEDICINAL CHEMISTRY, 1981, 24 (10) :1119-1124
[9]   MODE OF DEACTIVATION OF ENKEPHALINS BY RAT AND HUMAN-PLASMA AND RAT-BRAIN HOMOGENATES [J].
HAMBROOK, JM ;
MORGAN, BA ;
RANCE, MJ ;
SMITH, CFC .
NATURE, 1976, 262 (5571) :782-783
[10]  
HARTRODT B, 1982, PHARMAZIE, V37, P72
123