A-69024 - A NON-BENZAZEPINE ANTAGONIST WITH SELECTIVITY FOR THE DOPAMINE D-1 RECEPTOR

被引：38
作者：
KERKMAN, DJ
ACKERMAN, M
ARTMAN, LD
MACKENZIE, RG
JOHNSON, MC
BEDNARZ, L
MONTANA, W
ASIN, KE
STAMPFLI, H
KEBABIAN, JW
机构：
来源：
EUROPEAN JOURNAL OF PHARMACOLOGY | 1989年 / 166卷 / 03期
关键词：
D O I：
10.1016/0014-2999(89)90362-2
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：481 / 491
页数：11
相关论文
共 33 条
[1]   EVIDENCE FOR DIFFERENT STATES OF THE DOPAMINE D1 RECEPTOR - CLOZAPINE AND FLUPERLAPINE MAY PREFERENTIALLY LABEL AN ADENYLATE CYCLASE-COUPLED STATE OF THE D1-RECEPTOR [J].
ANDERSEN, PH ;
BRAESTRUP, C .
JOURNAL OF NEUROCHEMISTRY, 1986, 47 (06) :1822-1831
[2]   SOME ATYPICAL NEUROLEPTICS INHIBIT [H-3] SCH 23390 BINDING INVIVO [J].
ANDERSEN, PH ;
NIELSEN, EB ;
GRONVALD, FC ;
BRAESTRUP, C .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 120 (01) :143-144
[3]   DIFFERENTIAL INVOLVEMENT OF DOPAMINE D-1 AND D-2 RECEPTORS IN THE CIRCLING BEHAVIOR INDUCED BY APOMORPHINE, SK+F-38393, PERGOLIDE AND LY-171555 IN 6-HYDROXYDOPAMINE-LESIONED RATS [J].
ARNT, J ;
HYTTEL, J .
PSYCHOPHARMACOLOGY, 1985, 85 (03) :346-352
[4]   SYNTHESIS AND PHARMACOLOGICAL CHARACTERIZATION OF 1-PHENYL-1,2,3,4-TETRAHYDROISOQUINOLINE, 4-PHENYL-1,2,3,4-TETRAHYDROISOQUINOLINE, AND 1-BENZYL-1,2,3,4-TETRAHYDROISOQUINOLINE AS DOPAMINE RECEPTOR LIGANDS [J].
CHARIFSON, PS ;
WYRICK, SD ;
HOFFMAN, AJ ;
SIMMONS, RMA ;
BOWEN, JP ;
MCDOUGALD, DL ;
MAILMAN, RB .
JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (10) :1941-1946
[5]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[6]   PHARMACOLOGICAL EFFECTS OF A SPECIFIC DOPAMINE D-1 ANTAGONIST SCH-23390 IN COMPARISON WITH NEUROLEPTICS [J].
CHRISTENSEN, AV ;
ARNT, J ;
HYTTEL, J ;
LARSEN, JJ ;
SVENDSEN, O .
LIFE SCIENCES, 1984, 34 (16) :1529-1540
[7]   REVIEW - D1 DOPAMINE RECEPTOR - THE SEARCH FOR A FUNCTION - A CRITICAL-EVALUATION OF THE D1/D2 DOPAMINE RECEPTOR CLASSIFICATION AND ITS FUNCTIONAL IMPLICATIONS [J].
CLARK, D ;
WHITE, FJ .
SYNAPSE, 1987, 1 (04) :347-388
[8]   D-2 DOPAMINE RECEPTOR-MEDIATED INHIBITION OF ADENYLATE-CYCLASE ACTIVITY IN THE INTERMEDIATE LOBE OF THE RAT PITUITARY-GLAND REQUIRES GUANOSINE 5'-TRIPHOSPHATE [J].
COTE, TE ;
GREWE, CW ;
TSURUTA, K ;
STOOF, JC ;
ESKAY, RL ;
KEBABIAN, JW .
ENDOCRINOLOGY, 1982, 110 (03) :812-819
[9]   DOPAMINE-DERIVED ALKALOIDS IN ALCOHOLISM AND IN PARKINSONS AND HUNTINGTONS DISEASES [J].
DOSTERT, P ;
BENEDETTI, MS ;
DORDAIN, G .
JOURNAL OF NEURAL TRANSMISSION, 1988, 74 (02) :61-74
[10]   REGULATION OF AGONIST AND ANTAGONIST BINDING TO STRIATAL D-1 DOPAMINE-RECEPTORS - STUDIES USING THE SELECTIVE D-1 ANTAGONIST [H-3] SK-AND-F R-83566 [J].
FLAIM, KE ;
GESSNER, GW ;
CROOKE, ST ;
HEYS, JR ;
WEINSTOCK, J .
LIFE SCIENCES, 1986, 38 (23) :2087-2096
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