STRUCTURE OF THE HIGH-AFFINITY BINDING-SITE FOR NONCOMPETITIVE BLOCKERS OF THE ACETYLCHOLINE-RECEPTOR - SERINE-262 OF THE DELTA-SUBUNIT IS LABELED BY [H-3] CHLORPROMAZINE

被引：295

作者：

GIRAUDAT, J ^{[1
]}

DENNIS, M ^{[1
]}

HEIDMANN, T ^{[1
]}

CHANG, JY ^{[1
]}

CHANGEUX, JP ^{[1
]}

机构：

[1] CIBA GEIGY AG,PHARMACEUT RES LABS,CH-4002 BASEL,SWITZERLAND

来源：

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA | 1986年 / 83卷 / 08期

关键词：

D O I：

10.1073/pnas.83.8.2719

中图分类号：

O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];

学科分类号：

07 ; 0710 ; 09 ;

摘要：

引用

页码：2719 / 2723

页数：5

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COHEN, JB .

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[5]

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[6] ACETYLCHOLINE-RECEPTOR - AN ALLOSTERIC PROTEIN [J].

CHANGEUX, JP ;

DEVILLERSTHIERY, A ;

CHEMOUILLI, P .

SCIENCE, 1984, 225 (4668) :1335-1345

[7]

CHANGEUX JP, 1986, J PHYSL

[8] NUCLEOTIDE AND DEDUCED AMINO-ACID-SEQUENCES OF TORPEDO-CALIFORNICA ACETYLCHOLINE-RECEPTOR GAMMA-SUBUNIT [J].

CLAUDIO, T ;

BALLIVET, M ;

PATRICK, J ;

HEINEMANN, S .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (04) :1111-1115

[9]

COHEN JB, 1980, PROGR ANESTHESIOLOGY, V2, P165

[10]

DENNIS M, 1985, INT S MOL ASPECTS NE, P38

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