THE BENZODIAZEPINE GABA RECEPTOR COMPLEX - MOLECULAR-SIZE IN BRAIN SYNAPTIC-MEMBRANES AND IN SOLUTION

被引:69
作者
CHANG, LR [1 ]
BARNARD, EA [1 ]
机构
[1] UNIV LONDON IMPERIAL COLL SCI & TECHNOL,DEPT BIOCHEM,LONDON SW7 2AZ,ENGLAND
关键词
D O I
10.1111/j.1471-4159.1982.tb07983.x
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1507 / 1518
页数:12
相关论文
共 55 条
[1]   SOLUBLE GAMMA-AMINOBUTYRIC ACID AND BENZODIAZEPINE RECEPTORS FROM RAT CEREBRAL-CORTEX [J].
ASANO, T ;
OGASAWARA, N .
LIFE SCIENCES, 1981, 29 (02) :193-200
[2]   MUSCIMOL BINDING IN RAT-BRAIN - ASSOCIATION WITH SYNAPTIC GABA RECEPTORS [J].
BEAUMONT, K ;
CHILTON, WS ;
YAMAMURA, HI ;
ENNA, SJ .
BRAIN RESEARCH, 1978, 148 (01) :153-162
[3]   [H-3]-LABELED PROPYL BETA-CARBOLINE-3-CARBOXYLATE AS A SELECTIVE RADIOLIGAND FOR THE BZ1 BENZODIAZEPINE RECEPTOR SUBCLASS [J].
BRAESTRUP, C ;
NIELSEN, M .
JOURNAL OF NEUROCHEMISTRY, 1981, 37 (02) :333-341
[4]   PARTIAL AGONISTS FOR BRAIN GABA-BENZODIAZEPINE RECEPTOR COMPLEX [J].
BRAESTRUP, C ;
NIELSEN, M ;
KROGSGAARDLARSEN, P ;
FALCH, E .
NATURE, 1979, 280 (5720) :331-333
[5]  
BROWNER M, 1981, J NEUROSCI, V1, P514
[6]   MOLECULAR SIZES OF BENZODIAZEPINE RECEPTORS AND THE INTERACTING GABA RECEPTORS IN THE MEMBRANE ARE IDENTICAL [J].
CHANG, LR ;
BARNARD, EA ;
LO, MMS ;
DOLLY, JO .
FEBS LETTERS, 1981, 126 (02) :309-312
[7]   GABA RECEPTOR-MEDIATED MODULATION OF DIAZEPAM-H-3 BINDING IN RAT CORTEX [J].
CHIU, TH ;
ROSENBERG, HC .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 56 (04) :337-345
[8]   DIFFERENTIAL EFFECTS OF TRITON X-100 ON BENZODIAZEPINE AND GABA BINDING IN A FROZEN-THAWED SYNAPTOSOMAL FRACTION OF RAT-BRAIN [J].
CHIU, TH ;
ROSENBERG, HC .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 58 (03) :335-338
[9]   MOLECULAR MECHANISMS IN THE RECEPTOR ACTION OF BENZODIAZEPINES [J].
COSTA, E ;
GUIDOTTI, A .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1979, 19 :531-545
[10]   MOLECULAR-SIZE OF BENZODIAZEPINE RECEPTOR IN RAT-BRAIN INSITU - EVIDENCE FOR A FUNCTIONAL DIMER [J].
DOBLE, A ;
IVERSEN, LL .
NATURE, 1982, 295 (5849) :522-523