EFFECT OF MEMBRANE DEPOLARIZATION ON BINDING OF [NITRENDIPINE-H-3 TO RAT CARDIAC MYOCYTES

被引:71
作者
GREEN, FJ
FARMER, BB
WISEMAN, GL
JOSE, MJL
WATANABE, AM
机构
[1] INDIANA UNIV,SCH MED,DEPT MED,INDIANAPOLIS,IN 46202
[2] INDIANA UNIV,SCH MED,DEPT PHARMACOL,INDIANAPOLIS,IN 46202
关键词
D O I
10.1161/01.RES.56.4.576
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:576 / 585
页数:10
相关论文
共 48 条
[1]  
BELLEMANN P, 1981, ARZNEIMITTEL-FORSCH, V31-2, P2064
[2]   HIGH-AFFINITY BINDING OF A CALCIUM-CHANNEL ANTAGONIST TO SMOOTH AND CARDIAC-MUSCLE [J].
BOLGER, GT ;
GENGO, PJ ;
LUCHOWSKI, EM ;
SIEGEL, H ;
TRIGGLE, DJ ;
JANIS, RA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 104 (04) :1604-1609
[3]   CA-2+ CHANNEL MODULATION BY 8-BROMOCYCLIC AMP IN CULTURED HEART-CELLS [J].
CACHELIN, AB ;
DEPEYER, JE ;
KOKUBUN, S ;
REUTER, H .
NATURE, 1983, 304 (5925) :462-464
[4]  
CAMPBELL KP, 1983, J BIOL CHEM, V258, P1197
[5]  
CAMPBELL KP, 1984, J BIOL CHEM, V259, P5384
[6]  
CATTERALL WA, 1977, J BIOL CHEM, V252, P8669
[7]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[8]   [H-3] NIMODIPINE SPECIFIC BINDING TO CARDIAC MYOCYTES AND SUBCELLULAR-FRACTIONS [J].
DEPOVER, A ;
LEE, SW ;
MATLIB, MA ;
WHITMER, K ;
DAVIS, BA ;
POWELL, T ;
SCHWARTZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 113 (01) :185-191
[9]   SPECIFIC BINDING OF [H-3]LABELED NITRENDIPINE TO MEMBRANES FROM CORONARY-ARTERIES AND HEART IN RELATION TO PHARMACOLOGICAL EFFECTS - PARADOXICAL STIMULATION BY DILTIAZEM [J].
DEPOVER, A ;
MATLIB, MA ;
LEE, SW ;
DUBE, GP ;
GRUPP, IL ;
GRUPP, G ;
SCHWARTZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 108 (01) :110-117
[10]   DILTIAZEM POTENTIATES THE NEGATIVE INOTROPIC ACTION OF NIMODIPINE IN HEART [J].
DEPOVER, A ;
GRUPP, IL ;
GRUPP, G ;
SCHWARTZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1983, 114 (03) :922-929