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REVIEW - QUANTITATIVE STRUCTURE ACTIVITY RELATIONS BASED ON USE-DEPENDENT BLOCK AND REPRIMING KINETICS IN MYOCARDIUM
被引:72
|
作者
:
COURTNEY, KR
论文数:
0
引用数:
0
h-index:
0
COURTNEY, KR
机构
:
来源
:
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY
|
1987年
/ 19卷
/ 03期
关键词
:
D O I
:
10.1016/S0022-2828(87)80599-0
中图分类号
:
R5 [内科学];
学科分类号
:
1002 ;
100201 ;
摘要
:
引用
收藏
页码:319 / 330
页数:12
相关论文
共 27 条
[1]
THE CHARACTERIZATION OF SLOWER COMPONENT OF RECOVERY KINETICS FROM USE-DEPENDENT BLOCK ON SODIUM-CHANNEL WITH DISOPYRAMIDE
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HISATOME, I
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KINKI UNIV,OSAKA,JAPAN
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TAKAI, H
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KINKI UNIV,OSAKA,JAPAN
TAKAI, H
AIDA, Y
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MATSUNO, S
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KINKI UNIV,OSAKA,JAPAN
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KARASAKI, S
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KINKI UNIV,OSAKA,JAPAN
KARASAKI, S
OYAIZU, M
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0
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KINKI UNIV,OSAKA,JAPAN
OYAIZU, M
KOUMI, S
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0
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KINKI UNIV,OSAKA,JAPAN
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KATORI, R
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KINKI UNIV,OSAKA,JAPAN
KATORI, R
BIOPHYSICAL JOURNAL,
1993,
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[2]
Molecular determinants of mexiletine structure for potent and use-dependent block of skeletal muscle sodium channels
De Luca, A
论文数:
0
引用数:
0
h-index:
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Univ Bari, Fac Farm, Dipartimento Farmacobiol, Unita Farmacol, I-70125 Bari, Italy
De Luca, A
Natuzzi, F
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0
引用数:
0
h-index:
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机构:
Univ Bari, Fac Farm, Dipartimento Farmacobiol, Unita Farmacol, I-70125 Bari, Italy
Natuzzi, F
Desaphy, JF
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Farm, Dipartimento Farmacobiol, Unita Farmacol, I-70125 Bari, Italy
Desaphy, JF
Loni, G
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0
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0
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Univ Bari, Fac Farm, Dipartimento Farmacobiol, Unita Farmacol, I-70125 Bari, Italy
Loni, G
Lentini, G
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Univ Bari, Fac Farm, Dipartimento Farmacobiol, Unita Farmacol, I-70125 Bari, Italy
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Franchini, C
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Univ Bari, Fac Farm, Dipartimento Farmacobiol, Unita Farmacol, I-70125 Bari, Italy
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QUANTITATIVE-DETERMINATION OF RECOVERY KINETICS FROM USE-DEPENDENT DRUG UPTAKE - A TEST OF THE GUARDED RECEPTOR HYPOTHESIS
PACKER, DL
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DUKE UNIV,DURHAM,NC 27706
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GRANT, AO
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STRAUSS, HC
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STARMER, CF
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DUKE UNIV,DURHAM,NC 27706
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[4]
Specific mechanism of use-dependent channel block of calcium-permeable AMPA receptors provides activity-dependent inhibition of glutamatergic neurotransmission
Zaitsev, A. V.
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IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
Zaitsev, A. V.
Kim, K. K.
论文数:
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IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
Kim, K. K.
Fedorova, I. M.
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IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
Fedorova, I. M.
Dorofeeva, N. A.
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IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
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IM Sechenov Inst Evolutionary Physiol & Biochem R, St Petersburg 194223, Russia
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Termination of reentry by lidocaine in the tricuspid ring in vitro - Role of cycle-length oscillation, fast use-dependent kinetics, and fixed block
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[6]
EFFECTS OF RS-2135, A NEW ANTIARRHYTHMIC AGENT, ON THE KINETICS OF USE-DEPENDENT DECREASE IN MAXIMUM UPSTROKE VELOCITY IN GUINEA-PIG VENTRICULAR MYOCARDIUM
YORIKANE, R
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Use-dependent block of skeletal muscle sodium current by chiral derivatives of mexiletine and tocainide and antimyotonic activity on ADR mouse.
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Franchini, C
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[10]
Increased rigidity of the chiral centre of tocainide favours stereoselectivity and use-dependent block of skeletal muscle Na+ channels enhancing the antimyotonic activity in vivo
Talon, S
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Talon, S
De Luca, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
De Luca, A
De Bellis, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
De Bellis, M
Desaphy, JF
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0
引用数:
0
h-index:
0
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Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Desaphy, JF
Lentini, G
论文数:
0
引用数:
0
h-index:
0
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Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Lentini, G
Scilimati, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Scilimati, A
Corbo, F
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Corbo, F
Franchini, C
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Franchini, C
Tortorella, P
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Tortorella, P
Jockusch, H
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
Jockusch, H
Camerino, DC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Bari, Fac Pharm, Dept Pharmacobiol, Pharmacol Unit, I-70125 Bari, Italy
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134
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1531
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