TRANSFORMATIONS OF NITROPYRIMIDINES BY ACTION OF C-NUCLEOPHILES

被引：0

作者：

RUSINOV, VL ^{[1
]}

CHUPAKHIN, ON ^{[1
]}

VANDERPLAS, HC ^{[1
]}

机构：

[1] AGR UNIV WAGENINGEN,DEPT ORGAN CHEM,6803 BC WAGENINGEN,NETHERLANDS

来源：

HETEROCYCLES | 1995年 / 40卷 / 01期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The addition of C-nucleophiles to 5-nitropyrimidines, to some of their [1,5-a]pyrazolo- or triazolo-annelated systems, and their subsequent ring transformations have been reviewed. The ring transformations involving the replacement of the N-(3)-C-(4)-C-(5) fragment of the pyrimidine ring, the N-(1)-C-(5)-C-(6), the N-(1)-C-(2)-N-(3) or the N-(1)-C-(2) fragment by structural parts of different C-nucleophilic agents are summarized; possible pathways, involving these transformations are discussed.

引用

页码：441 / 475

页数：35

共 52 条

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