INTERACTION OF ARYLPIPERAZINES WITH 5-HT1A, 5-HT1B, 5-HT1C AND 5-HT1D RECEPTORS - DO DISCRIMINATORY 5-HT1B RECEPTOR LIGANDS EXIST

被引:0
作者
SCHOEFFTER, P [1 ]
HOYER, D [1 ]
机构
[1] SANDOZ LTD,PRECLIN RES,BLDG 386-521,CH-4002 BASEL,SWITZERLAND
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:675 / 683
页数:9
相关论文
共 53 条
[1]   5-HT-1A AND 5-HT-1B SELECTIVITY OF 2 PHENYLPIPERAZINE DERIVATIVES - EVIDENCE FOR 5-HT-1B HETEROGENEITY [J].
ASARCH, KB ;
RANSOM, RW ;
SHIH, JC .
LIFE SCIENCES, 1985, 36 (13) :1265-1273
[2]  
BOCKAERT J, 1987, N-S ARCH PHARMACOL, V335, P588
[3]   5-HT1B RECEPTORS ARE NEGATIVELY COUPLED WITH ADENYLATE-CYCLASE IN RAT SUBSTANTIA NIGRA [J].
BOUHELAL, R ;
SMOUNYA, L ;
BOCKAERT, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 151 (02) :189-196
[4]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[5]   A UNIQUE SEROTONIN RECEPTOR IN CHOROID-PLEXUS IS LINKED TO PHOSPHATIDYLINOSITOL TURNOVER [J].
CONN, PJ ;
SANDERSBUSH, E ;
HOFFMAN, BJ ;
HARTIG, PR .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (11) :4086-4088
[6]  
CONN PJ, 1987, J PHARMACOL EXP THER, V242, P552
[7]  
CORTES R, 1984, BRIT J PHARMACOL, V81, pP202
[8]  
DELEAN A, 1980, J BIOL CHEM, V255, P7108
[9]  
DEVIVO M, 1986, J PHARMACOL EXP THER, V238, P248
[10]   INHIBITION OF FORSKOLIN-STIMULATED ADENYLATE-CYCLASE ACTIVITY BY 5-HT RECEPTOR AGONISTS [J].
DEVIVO, M ;
MAAYANI, S .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 119 (03) :231-234