POTASSIUM CHANNEL ACTIVATOR DRUGS - MECHANISM OF ACTION, PHARMACOLOGICAL PROPERTIES, AND THERAPEUTIC POTENTIAL

被引:151
作者
LONGMAN, SD
HAMILTON, TC
机构
[1] SmithKline Beecham Pharmaceuticals, Medicinal Research Centre, Harlow, Essex, Coldharbour Road
关键词
D O I
10.1002/med.2610120202
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:73 / 148
页数:76
相关论文
共 524 条
[21]   GLUCOSE INDUCES CLOSURE OF SINGLE POTASSIUM CHANNELS IN ISOLATED RAT PANCREATIC BETA-CELLS [J].
ASHCROFT, FM ;
HARRISON, DE ;
ASHCROFT, SJH .
NATURE, 1984, 312 (5993) :446-448
[22]  
ASHCROFT FM, 1988, ANNU REV NEUROSCI, V11, P97, DOI 10.1146/annurev.ne.11.030188.000525
[23]   ADENOSINE-5'-TRIPHOSPHATE-SENSITIVE ION CHANNELS IN NEONATAL RAT CULTURED CENTRAL NEURONS [J].
ASHFORD, MLJ ;
STURGESS, NC ;
TROUT, NJ ;
GARDNER, NJ ;
HALES, CN .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1988, 412 (03) :297-304
[24]   GLUCOSE-INDUCED EXCITATION OF HYPOTHALAMIC NEURONS IS MEDIATED BY ATP-SENSITIVE K+ CHANNELS [J].
ASHFORD, MLJ ;
BODEN, PR ;
TREHERNE, JM .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1990, 415 (04) :479-483
[25]  
ASHFORD MLJ, 1989, J PHYSL, V409, pP53
[26]   POTASSIUM CHANNEL BLOCKADE - A MECHANISM FOR SUPPRESSING VENTRICULAR-FIBRILLATION [J].
BACANER, MB ;
CLAY, JR ;
SHRIER, A ;
BROCHU, RM .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (07) :2223-2227
[27]   EFFECT OF PINACIDIL ON MYOCARDIAL BLOOD-FLOW IN THE PRESENCE OF A CORONARY-ARTERY STENOSIS [J].
BACHE, RJ ;
DAI, XZ ;
BARAN, KW .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1990, 15 (04) :618-625
[28]  
BAIRD A, 1988, BRIT J CLIN PHARMACO, V25, pP114
[29]   MEMBRANE HYPERPOLARIZATION, CYCLIC-NUCLEOTIDE LEVELS AND RELAXATION IN THE GUINEA-PIG INTERNAL ANAL-SPHINCTER [J].
BAIRD, AA ;
MUIR, TC .
BRITISH JOURNAL OF PHARMACOLOGY, 1990, 100 (02) :329-335
[30]   CLINICAL PHARMACOKINETICS OF SULFONYLUREA HYPOGLYCEMIC DRUGS [J].
BALANT, L .
CLINICAL PHARMACOKINETICS, 1981, 6 (03) :215-241