NUCLEOTIDE INTERACTIONS WITH 5-HT1A BINDING-SITES DIRECTLY LABELED BY [H-3] 8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN ([H-3]-8-OH-DPAT)

被引:91
作者
SCHLEGEL, JR [1 ]
PEROUTKA, SJ [1 ]
机构
[1] STANFORD UNIV,MED CTR,DEPT NEUROL,STANFORD,CA 94305
关键词
D O I
10.1016/0006-2952(86)90725-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1943 / 1949
页数:7
相关论文
共 39 条
[11]   ALPHA-NORADRENERGIC RECEPTORS IN BRAIN MEMBRANES - SODIUM, MAGNESIUM AND GUANYL NUCLEOTIDES MODULATE AGONIST BINDING [J].
GLOSSMANN, H ;
PRESEK, P .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 306 (01) :67-73
[12]   IDENTIFICATION OF PRE-SYNAPTIC SEROTONIN AUTORECEPTORS USING A NEW LIGAND - H-3-PAT [J].
GOZLAN, H ;
ELMESTIKAWY, S ;
PICHAT, L ;
GLOWINSKI, J ;
HAMON, M .
NATURE, 1983, 305 (5930) :140-142
[13]   [H-3]8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN BINDING TO PRESYNAPTIC AND POSTSYNAPTIC 5-HYDROXYTRYPTAMINE SITES IN VARIOUS REGIONS OF THE RAT-BRAIN [J].
HALL, MD ;
ELMESTIKAWY, S ;
EMERIT, MB ;
PICHAT, L ;
HAMON, M ;
GOZLAN, H .
JOURNAL OF NEUROCHEMISTRY, 1985, 44 (06) :1685-1696
[14]   BIOCHEMICAL-EVIDENCE FOR THE 5-HT AGONIST PROPERTIES OF PAT (8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN) IN THE RAT-BRAIN [J].
HAMON, M ;
BOURGOIN, S ;
GOZLAN, H ;
HALL, MD ;
GOETZ, C ;
ARTAUD, F ;
HORN, AS .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 100 (3-4) :263-276
[15]  
HAMON M, 1984, HDB NEUROCHEMISTRY, V6, P107
[16]  
LEFKOWITZ RJ, 1976, J BIOL CHEM, V251, P4686
[17]  
LIMBIRD LE, 1981, BIOCHEM J, V195, P1
[18]  
MAGUIRE ME, 1976, MOL PHARMACOL, V12, P335
[19]   CA-2(+)-GUANINE NUCLEOTIDE INTERACTIONS IN BRAIN MEMBRANES .1. MODULATION OF CENTRAL 5-HYDROXYTRYPTAMINE RECEPTORS IN THE RAT [J].
MALLAT, M ;
HAMON, M .
JOURNAL OF NEUROCHEMISTRY, 1982, 38 (01) :151-161
[20]   AUTORADIOGRAPHIC EVIDENCE FOR THE HETEROGENEITY OF 5-HT1 SITES IN THE RAT-BRAIN [J].
MARCINKIEWICZ, M ;
VERGE, D ;
GOZLAN, H ;
PICHAT, L ;
HAMON, M .
BRAIN RESEARCH, 1984, 291 (01) :159-163