NUCLEOTIDE INTERACTIONS WITH 5-HT1A BINDING-SITES DIRECTLY LABELED BY [H-3] 8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN ([H-3]-8-OH-DPAT)

被引:91
作者
SCHLEGEL, JR [1 ]
PEROUTKA, SJ [1 ]
机构
[1] STANFORD UNIV,MED CTR,DEPT NEUROL,STANFORD,CA 94305
关键词
D O I
10.1016/0006-2952(86)90725-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1943 / 1949
页数:7
相关论文
共 39 条
[1]   SEROTONIN-ELICITED AMPLIFICATION OF ADENYLATE-CYCLASE ACTIVITY IN HIPPOCAMPAL MEMBRANES FROM ADULT-RAT [J].
BARBACCIA, ML ;
BRUNELLO, N ;
CHUANG, DM ;
COSTA, E .
JOURNAL OF NEUROCHEMISTRY, 1983, 40 (06) :1671-1679
[2]   GUANYL NUCLEOTIDE AND DIVALENT-CATION REGULATION OF CORTICAL-S2 SEROTONIN RECEPTORS [J].
BATTAGLIA, G ;
SHANNON, M ;
TITELER, M .
JOURNAL OF NEUROCHEMISTRY, 1984, 43 (05) :1213-1219
[3]  
Bockaert J, 1981, Adv Exp Med Biol, V133, P327
[4]  
CREESE I, 1979, MOL PHARMACOL, V16, P69
[5]   H-3-TVX Q-7821 - IDENTIFICATION OF 5-HT1 BINDING-SITES AS TARGET FOR A NOVEL PUTATIVE ANXIOLYTIC [J].
DOMPERT, WU ;
GLASER, T ;
TRABER, J .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 328 (04) :467-470
[6]  
Fillion G, 1983, J Neural Transm Suppl, V18, P307
[7]   DECREASE OF [5-HT-H-3 HIGH-AFFINITY BINDING AND 5-HT ADENYLATE-CYCLASE ACTIVATION AFTER KAINIC ACID LESION IN RAT-BRAIN STRIATUM [J].
FILLION, G ;
BEAUDOIN, D ;
ROUSSELLE, JC ;
DENIAU, JM ;
FILLION, MP ;
DRAY, F ;
JACOB, J .
JOURNAL OF NEUROCHEMISTRY, 1979, 33 (02) :567-570
[8]  
FILLION G, 1979, LIFE SCI, V24, P1813, DOI 10.1016/0024-3205(79)90072-9
[9]  
FILLION GMB, 1978, MOL PHARMACOL, V14, P50
[10]   G-PROTEINS AND DUAL CONTROL OF ADENYLATE-CYCLASE [J].
GILMAN, AG .
CELL, 1984, 36 (03) :577-579