STRUCTURE - ACTIVITY RELATIONSHIP STUDIES OF COCAINE - REPLACEMENT OF THE C-2 ESTER GROUP BY VINYL ARGUES AGAINST H-BONDING AND PROVIDES AN ESTERASE-RESISTANT, HIGH-AFFINITY COCAINE ANALOG

被引：70

作者：

KOZIKOWSKI, AP ^{[1
]}

ROBERTI, M ^{[1
]}

XIANG, L ^{[1
]}

BERGMANN, JS ^{[1
]}

CALLAHAN, PM ^{[1
]}

CUNNINGHAM, KA ^{[1
]}

JOHNSON, KM ^{[1
]}

机构：

[1] UNIV TEXAS,MED BRANCH,DEPT PHARMACOL & TOXICOL,GALVESTON,TX 77555

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1992年 / 35卷 / 25期

关键词：

D O I：

10.1021/jm00103a015

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：4764 / 4766

页数：3

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