STRUCTURE-BASED DESIGN OF HIV-1 PROTEASE INHIBITORS - REPLACEMENT OF 2 AMIDES AND A 10-PI-AROMATIC SYSTEM BY A FUSED BIS-TETRAHYDROFURAN

被引：63

作者：

GHOSH, AK

THOMPSON, WJ

FITZGERALD, PMD

CULBERSON, JC

AXEL, MG

MCKEE, SP

HUFF, JR

ANDERSON, PS

机构：

[1] MERCK SHARP & DOHME LTD,RES LABS,DEPT MED CHEM,W POINT,PA 19486

[2] MERCK SHARP & DOHME LTD,RES LABS,DEPT BIOPHYS CHEM,W POINT,PA 19486

[3] MERCK SHARP & DOHME LTD,RES LABS,DEPT MOLEC SYST,W POINT,PA 19486

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1994年 / 37卷 / 16期

关键词：

D O I：

10.1021/jm00042a002

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：2506 / 2508

页数：3

共 13 条

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