TACHYKININ ANTAGONISTS HAVE POTENT LOCAL-ANESTHETIC ACTIONS

被引:69
作者
POST, C
BUTTERWORTH, JF
STRICHARTZ, GR
KARLSSON, JA
PERSSON, CGA
机构
[1] AB DRACO,DEPT RES & DEV,BOX 34,S-22100 LUND,SWEDEN
[2] ASTRA LAKEMEDEL AB,RES & DEV LABS,S-15185 SODERTALJE,SWEDEN
[3] UNIV LUND,DEPT CLIN PHARMACOL,S-22101 LUND,SWEDEN
[4] HARVARD UNIV,BRIGHAM & WOMENS HOSP,SCH MED,ANESTHESIA RES LAB,BOSTON,MA 02115
关键词
D O I
10.1016/0014-2999(85)90008-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:347 / 354
页数:8
相关论文
共 32 条
[1]   INTRATHECAL (D-PRO2,D-TRP7,9)-SP ELICITS HYPOALGESIA AND MOTOR BLOCKADE IN THE RAT AND ANTAGONIZES NOXIOUS RESPONSES INDUCED BY SUBSTANCE-P [J].
AKERMAN, B ;
ROSELL, S ;
FOLKERS, K .
ACTA PHYSIOLOGICA SCANDINAVICA, 1982, 114 (04) :631-633
[2]  
BOIVIE J, 1975, MTP INT REV SCIENC 1, V3, P303
[3]  
COURTNEY KR, 1978, ANESTHESIOLOGY, V48, P11
[4]   A SYNTHETIC PEPTIDE AS AN ANTAGONIST OF SUBSTANCE-P [J].
ENGBERG, G ;
SVENSSON, TH ;
ROSELL, S ;
FOLKERS, K .
NATURE, 1981, 293 (5829) :222-223
[5]  
ERLANGER J, 1937, ELECTRICAL SIGNS NER
[6]   DIFFERENTIAL SENSITIVITIES OF MAMMALIAN NERVE-FIBERS TO LOCAL-ANESTHETIC AGENTS [J].
GISSEN, AJ ;
COVINO, BG ;
GREGUS, J .
ANESTHESIOLOGY, 1980, 53 (06) :467-474
[7]   3 TACHYKININS IN MAMMALIAN BRAIN [J].
HARMAR, AJ .
TRENDS IN NEUROSCIENCES, 1984, 7 (03) :57-60
[8]   IMMUNOHISTOCHEMICAL EVIDENCE FOR A NEUROTOXIC ACTION OF (D-PRO2,D-TRP7,9)-SUBSTANCE-P, AN ANALOG WITH SUBSTANCE-P ANTAGONISTIC ACTIVITY [J].
HOKFELT, T ;
VINCENT, S ;
HELLSTEN, L ;
ROSELL, S ;
FOLKERS, K ;
MARKEY, K ;
GOLDSTEIN, M ;
CUELLO, C .
ACTA PHYSIOLOGICA SCANDINAVICA, 1981, 113 (04) :571-573
[9]   A SUBSTANCE-P ANTAGONIST, [D-PRO2, D-TRP7,9]SP, INHIBITS INFLAMMATORY RESPONSES IN THE RABBIT EYE [J].
HOLMDAHL, G ;
HAKANSON, R ;
LEANDER, S ;
ROSELL, S ;
FOLKERS, K ;
SUNDLER, F .
SCIENCE, 1981, 214 (4524) :1029-1031
[10]   LOCAL-ANESTHETICS SELECTIVELY INHIBIT NON-CHOLINERGIC NEURAL CONTRACTIONS IN GUINEA-PIG AIRWAYS [J].
KARLSSON, JA ;
PERSSON, CGA .
ACTA PHYSIOLOGICA SCANDINAVICA, 1984, 120 (03) :469-471