THE DESIGN, SYNTHESIS, AND CHARACTERIZATION OF TIGHT-BINDING INHIBITORS OF CALMODULIN

被引：65
作者：
DEGRADO, WF
PRENDERGAST, FG
WOLFE, HR
COX, JA
机构：
[1] MAYO CLIN & MAYO FDN, DEPT PHARMACOL, ROCHESTER, MN 55901 USA
[2] UNIV GENEVA, DEPT BIOCHEM, CH-1211 GENEVA 4, SWITZERLAND
来源：
JOURNAL OF CELLULAR BIOCHEMISTRY | 1985年 / 29卷 / 02期
关键词：
D O I：
10.1002/jcb.240290204
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：83 / 93
页数：11
相关论文
共 33 条
[1]   3-DIMENSIONAL STRUCTURE OF CALMODULIN [J].
BABU, YS ;
SACK, JS ;
GREENHOUGH, TJ ;
BUGG, CE ;
MEANS, AR ;
COOK, WJ .
NATURE, 1985, 315 (6014) :37-40
[2]  
BARANY G, 1980, PEPTIDES, V2, P3
[3]  
BLUMENTHAL DK, 1985, BIOPHYS J, V47, pA76
[4]  
CANTOR CR, 1981, BIOPHYSICAL CHEM 3, P1041
[5]   DETERMINATION OF HELIX AND BETA-FORM OF PROTEINS IN AQUEOUS-SOLUTION BY CIRCULAR-DICHROISM [J].
CHEN, YH ;
YANG, JT ;
CHAU, KH .
BIOCHEMISTRY, 1974, 13 (16) :3350-3359
[6]   CA2+-DEPENDENT HIGH-AFFINITY COMPLEX-FORMATION BETWEEN CALMODULIN AND MELITTIN [J].
COMTE, M ;
MAULET, Y ;
COX, JA .
BIOCHEMICAL JOURNAL, 1983, 209 (01) :269-272
[7]  
COX JA, 1985, J BIOL CHEM, V260, P2527
[8]   SOLID-PHASE SYNTHESIS OF PROTECTED PEPTIDES ON A POLYMER-BOUND OXIME - PREPARATION OF SEGMENTS COMPRISING THE SEQUENCE OF A CYTO-TOXIC 26-PEPTIDE ANALOG [J].
DEGRADO, WF ;
KAISER, ET .
JOURNAL OF ORGANIC CHEMISTRY, 1982, 47 (17) :3258-3261
[9]   IDENTIFICATION OF BETA-ENDORPHIN RESIDUES 14-25 AS A REGION INVOLVED IN THE INHIBITION OF CALMODULIN-STIMULATED PHOSPHODIESTERASE ACTIVITY [J].
GIEDROC, DP ;
LING, N ;
PUETT, D .
BIOCHEMISTRY, 1983, 22 (24) :5584-5591
[10]   FUNCTIONAL-PROPERTIES OF COVALENT BETA-ENDORPHIN PEPTIDE CALMODULIN COMPLEXES - CHLORPROMAZINE BINDING AND PHOSPHODIESTERASE ACTIVATION [J].
GIEDROC, DP ;
KERAVIS, TM ;
STAROS, JV ;
LING, N ;
WELLS, JN ;
PUETT, D .
BIOCHEMISTRY, 1985, 24 (05) :1203-1211
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