CONFORMATIONALLY CONSTRAINED AMINO-ACIDS - SYNTHESIS OF NOVEL 3,4-CYCLIZED TRYPTOPHANS

被引：15
|
作者：
HORWELL, DC [1 ]
NICHOLS, PD [1 ]
ROBERTS, E [1 ]
机构：
[1] ADDENBROOKES HOSP,PARKE DAVIS NEUROSCI RES CTR,CAMBRIDGE CB2 2QB,ENGLAND
来源：
TETRAHEDRON LETTERS | 1994年 / 35卷 / 06期
关键词：
CONFORMATIONAL; TRYPTOPHAN; 3,4-CYCLIZATION; SYNTHESIS; HECK;
D O I：
10.1016/S0040-4039(00)76005-9
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The synthesis of novel conformationally constrained tryptophan derivatives via a Heck-type cyclisation of an unusual alpha-substituted amino acid is described.
引用
收藏
页码：939 / 940
页数：2
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