CONFORMATIONALLY CONSTRAINED AMINO-ACIDS - SYNTHESIS OF NOVEL 3,4-CYCLIZED TRYPTOPHANS

被引：15

作者：

HORWELL, DC ^{[1
]}

NICHOLS, PD ^{[1
]}

ROBERTS, E ^{[1
]}

机构：

[1] ADDENBROOKES HOSP,PARKE DAVIS NEUROSCI RES CTR,CAMBRIDGE CB2 2QB,ENGLAND

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 06期

关键词：

CONFORMATIONAL; TRYPTOPHAN; 3,4-CYCLIZATION; SYNTHESIS; HECK;

D O I：

10.1016/S0040-4039(00)76005-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of novel conformationally constrained tryptophan derivatives via a Heck-type cyclisation of an unusual alpha-substituted amino acid is described.

引用

页码：939 / 940

页数：2

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