WIDESPREAD DISTRIBUTION OF BRAIN DOPAMINE-RECEPTORS EVIDENCED WITH [I-125]IODOSULPRIDE, A HIGHLY SELECTIVE LIGAND

被引:257
作者
MARTRES, MP [1 ]
BOUTHENET, ML [1 ]
SALES, N [1 ]
SOKOLOFF, P [1 ]
SCHWARTZ, JC [1 ]
机构
[1] FAC PHARM PARIS,F-75270 PARIS 06,FRANCE
关键词
D O I
10.1126/science.3838821
中图分类号
O [数理科学和化学]; P [天文学、地球科学]; Q [生物科学]; N [自然科学总论];
学科分类号
07 ; 0710 ; 09 ;
摘要
引用
收藏
页码:752 / 755
页数:4
相关论文
共 42 条
[1]   BETA-ADRENERGIC-RECEPTOR - STEREOSPECIFIC INTERACTION OF IODINATED BETA-BLOCKING AGENT WITH HIGH AFFINITY SITE [J].
AURBACH, GD ;
FEDAK, SA ;
WOODARD, CJ ;
PALMER, JS .
SCIENCE, 1974, 186 (4170) :1223-1224
[2]   EFFERENT CONNECTIONS OF THE SUBSTANTIA NIGRA AND VENTRAL TEGMENTAL AREA IN THE RAT [J].
BECKSTEAD, RM ;
DOMESICK, VB ;
NAUTA, WJH .
BRAIN RESEARCH, 1979, 175 (02) :191-217
[3]   DOPAMINERGIC INNERVATION OF RAT PREFRONTAL CORTEX - FLUORESCENCE HISTOCHEMICAL STUDY [J].
BERGER, B ;
THIERRY, AM ;
TASSIN, JP ;
MOYNE, MA .
BRAIN RESEARCH, 1976, 106 (01) :133-145
[4]   BIOCHEMICAL-EVIDENCE FOR A TRANSMITTER ROLE OF DOPAMINE IN THE RAT HIPPOCAMPUS [J].
BISCHOFF, S ;
SCATTON, B ;
KORF, J .
BRAIN RESEARCH, 1979, 165 (01) :161-165
[5]  
BOUTHENET ML, UNPUB
[6]   DIRECT ROLE OF DOPAMINE IN THE RAT SUBTHALAMIC NUCLEUS AND AN ADJACENT INTRAPEDUNCULAR AREA [J].
BROWN, LL ;
MAKMAN, MH ;
WOLFSON, LI ;
DVORKIN, B ;
WARNER, C ;
KATZMAN, R .
SCIENCE, 1979, 206 (4425) :1416-1418
[7]   A RAPID FILTRATION ASSAY FOR SOLUBLE RECEPTORS USING POLYETHYLENIMINE-TREATED FILTERS [J].
BRUNS, RF ;
LAWSONWENDLING, K ;
PUGSLEY, TA .
ANALYTICAL BIOCHEMISTRY, 1983, 132 (01) :74-81
[8]   PREPARATION OF N(1-ETHYL-2-PYRROLIDYL-METHYL)2-METHOXY-4-IODO-I-125-5-ETHYL SULFONYL BENZAMIDE - A RADIOLIGAND FOR THE RADIOIMMUNOASSAY OF SULPIRIDE-RELATED COMPOUNDS [J].
CARDOSO, MT ;
PRADELLES, P .
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1982, 19 (09) :1103-1109
[9]   DOPAMINE RECEPTOR-BINDING PREDICTS CLINICAL AND PHARMACOLOGICAL POTENCIES OF ANTI-SCHIZOPHRENIC DRUGS [J].
CREESE, I ;
BURT, DR ;
SNYDER, SH .
SCIENCE, 1976, 192 (4238) :481-483
[10]   DISTRIBUTION OF PUTATIVE NEUROTRANSMITTERS IN THE NEOCORTEX [J].
EMSON, PC ;
LINDVALL, O .
NEUROSCIENCE, 1979, 4 (01) :1-30