SYNTHESIS AND INHIBITING ACTIVITY OF PEPTIDYLKETONES AS SUBSTRATE-ANALOGS OF PAPAIN

被引：14

作者：

GIORDANO, C

GALLINA, C

CONSALVI, V

SCANDURRA, R

机构：

[1] UNIV ROME LA SAPIENZA,DIPARTIMENTO STUDI FARMACEUT,PLE A MORO 5,I-00185 ROME,ITALY

[2] UNIV ROME LA SAPIENZA,DIPARTIMENTO STUDI FARMACEUT,I-00185 ROME,ITALY

[3] UNIV ROME LA SAPIENZA,CNR,CTR STUDIO CHIM FARM,I-00185 ROME,ITALY

来源：

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | 1989年 / 24卷 / 04期

关键词：

D O I：

10.1016/0223-5234(89)90078-0

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：357 / 362

页数：6

共 37 条

[1]

ARNDT F, 1932, MONATSH CHEM, V59, P215

[2]

Bell R. P., 1966, ADV PHYS ORG CHEM, P1, DOI DOI 10.1016/S0065-3160(08)60351-2

[3] REACTIONS OF PAPAIN AND OF LOW-MOLECULAR-WEIGHT THIOLS WITH SOME AROMATIC DISULFIDES - 2,2'-DIPYRIDYL DISULFIDE AS A CONVENIENT ACTIVE-SITE TITRANT FOR PAPAIN EVEN IN PRESENCE OF OTHER THIOLS [J].

BROCKLEHURST, K ;

LITTLE, G .

BIOCHEMICAL JOURNAL, 1973, 133 (01) :67-80

[4] TIGHT-BINDING INHIBITORS .1. KINETIC-BEHAVIOR [J].

CHA, S .

BIOCHEMICAL PHARMACOLOGY, 1975, 24 (23) :2177-2185

[5]

CHA S, 1976, BIOCHEM PHARMACOL, V25, P1561

[6]

CHEN FM, 1983, J ORG CHEM, V26, P2939

[7] TRICHLOROAMINOALCOHOLS .1. 1,1,1-TRICHLORO-3-AMINOPROPANOL-2 AND DERIVATIVES [J].

COMPTON, M ;

HIGGINS, H ;

MACBETH, L ;

OSBORN, J ;

BURKETT, H .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1949, 71 (09) :3229-3231

[8] THE PREPARATION AND REACTIONS OF SOME FLUORINE-CONTAINING NITRO COMPOUNDS [J].

COOK, DJ ;

PIERCE, OR ;

MCBEE, ET .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1954, 76 (01) :83-87

[9] REVERSIBLE, SLOW, TIGHT-BINDING INHIBITION OF HUMAN-LEUKOCYTE ELASTASE [J].

DUNLAP, RP ;

STONE, PJ ;

ABELES, RH .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1987, 145 (01) :509-513

[10] BIOLOGICALLY ORIENTED ORGANIC SULFUR CHEMISTRY .I. REACTIONS OF THIOLS WITH HIGHLY REACTIVE CARBONYL COMPOUNDS [J].

FIELD, L ;

SWEETMAN, BJ .

JOURNAL OF ORGANIC CHEMISTRY, 1969, 34 (06) :1799-&

← 1 2 3 4 →