SODIUM-IONS INCREASE THE BINDING OF THE ANTAGONIST PEPTIDE ICI-174864 TO THE DELTA-OPIATE RECEPTOR

被引:18
作者
APPELMANS, N
CARROLL, JA
RANCE, MJ
SIMON, EJ
TRAYNOR, JR
机构
[1] LOUGHBOROUGH UNIV TECHNOL,DEPT CHEM,LOUGHBOROUGH LE11 3TU,LEICS,ENGLAND
[2] NYU MED CTR,DEPT PSYCHIAT & PHARMACOL,NEW YORK,NY 10016
[3] ICI PLC,DIV PHARMACEUT,DEPT BIOSCI 2,MACCLESFIELD SK10 4TG,CHESHIRE,ENGLAND
关键词
D O I
10.1016/0143-4179(86)90089-2
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:139 / 143
页数:5
相关论文
共 8 条
[1]   MU-RECEPTOR BINDING IN PHYSIOLOGICAL MEDIA - COMPARISON WITH ISOLATED TISSUE DATA [J].
CARROLL, JA ;
MILLER, L ;
SHAW, JS ;
DOWNES, CP .
NEUROPEPTIDES, 1984, 5 (1-3) :89-92
[2]   SELECTIVITIES OF OPIOID PEPTIDE ANALOGS AS AGONISTS AND ANTAGONISTS AT THE DELTA-RECEPTOR [J].
CORBETT, AD ;
GILLAN, MGC ;
KOSTERLITZ, HW ;
MCKNIGHT, AT ;
PATERSON, SJ ;
ROBSON, LE .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (01) :271-279
[3]   ICI-174864 - A HIGHLY SELECTIVE ANTAGONIST FOR THE OPIOID DELTA-RECEPTOR [J].
COTTON, R ;
GILES, MG ;
MILLER, L ;
SHAW, JS ;
TIMMS, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 97 (3-4) :331-332
[4]   THE USE OF [H-3]-[D-PEN2,D-PEN5]ENKEPHALIN AS A HIGHLY SELECTIVE LIGAND FOR THE DELTA-BINDING SITE [J].
COTTON, R ;
KOSTERLITZ, HW ;
PATERSON, SJ ;
RANCE, MJ ;
TRAYNOR, JR .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (04) :927-932
[5]   NEUROBLASTOMA X GLIOMA HYBRID CELL LINE WITH MORPHINE RECEPTORS [J].
KLEE, WA ;
NIRENBER.M .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1974, 71 (09) :3474-3477
[6]  
PERT CB, 1974, MOL PHARMACOL, V10, P868
[7]   SOLUBILIZATION OF A STEREOSPECIFIC OPIATE-MACROMOLECULAR COMPLEX FROM RAT-BRAIN [J].
SIMON, EJ ;
HILLER, JM ;
EDELMAN, I .
SCIENCE, 1975, 190 (4212) :389-390
[8]  
SIMON EJ, 1975, J PHARMACOL EXP THER, V192, P531