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- [1] MCC950 closes the active conformation of NLRP3 to an inactive stateNature Chemical Biology, 2019, 15 : 560 - 564Ana Tapia-Abellán论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBDiego Angosto-Bazarra论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBHelios Martínez-Banaclocha论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBCarlos de Torre-Minguela论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBJose P. Cerón-Carrasco论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBHoracio Pérez-Sánchez论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBJuan I. Arostegui论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBPablo Pelegrin论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIB
- [2] MCC950 closes the active conformation of NLRP3 to an inactive stateNATURE CHEMICAL BIOLOGY, 2019, 15 (06) : 560 - +Tapia-Abelian, Ana论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, SpainAngosto-Bazarra, Diego论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, SpainMartinez-Banaclocha, Helios论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spainde Torre-Minguela, Carlos论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, SpainCeron-Carrasco, Jose P.论文数: 0 引用数: 0 h-index: 0机构: Univ Catolica Murcia UCAM, Comp Engn Dept, Bioinformat & High Performance Comp Res Grp BIO H, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, SpainPerez-Sanchez, Horacio论文数: 0 引用数: 0 h-index: 0机构: Univ Catolica Murcia UCAM, Comp Engn Dept, Bioinformat & High Performance Comp Res Grp BIO H, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, SpainArostegui, Juan, I论文数: 0 引用数: 0 h-index: 0机构: Hosp Clin IDIBAPS, Dept Immunol, Barcelona, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, SpainPelegrin, Pablo论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spain Univ Clin Hosp Virgen de la Arrixaca, Biomed Res Inst Murcia IMIB Arrixaca, Murcia, Spain
- [3] MCC950 closes the active conformation of NLRP3 to an inactive state (vol 15, pg 560, 2019)NATURE CHEMICAL BIOLOGY, 2021, 17 (03) : 361 - 361Tapia-Abellan, Ana论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBAngosto-Bazarra, Diego论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBMartinez-Banaclocha, Helios论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBde Torre-Minguela, Carlos论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBCeron-Carrasco, Jose P.论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBPerez-Sanchez, Horacio论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBArostegui, Juan I.论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIBPelegrin, Pablo论文数: 0 引用数: 0 h-index: 0机构: University Clinical Hospital Virgen de la Arrixaca,Biomedical Research Institute of Murcia (IMIB
- [4] Integrated Proteomics Characterization of NLRP3 Inflammasome Inhibitor MCC950 in Monocytic Cell Line Confirms Direct MCC950 Engagement with Endogenous NLRP3ACS CHEMICAL BIOLOGY, 2024, 19 (04) : 962 - 972Zhao, Heng论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USAKumar, Praveen论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Quantitat Biol, Discovery Sci, R&D, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USASobreira, Tiago Jose Paschoal论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Quantitat Biol, Discovery Sci, R&D, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USASmith, Mackenzie论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USANovick, Steven论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Quantitat Biol, Discovery Sci, R&D, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USAJohansson, Anders论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Med Chem Res & Early Dev, Cardiovasc Renal & Metab CVRM, BioPharmaceut R&D, Gothenburg, Sweden AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USALuchniak, Anna论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Mechanist & Struct Biol, Discovery Sci, R&D, S-43183 Gothenburg, Sweden AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USAZhang, Andrew论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USAWoollard, Kevin J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Biosci Renal Res & Early Dev, Cardiovasc Renal & Metab CVRM, BioPharmaceut R&D, Cambridge CB2 OAA, England AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USALarsson, Niklas论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Biol, Discovery Sci, R&D, S-43183 Gothenburg, Sweden AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USAKawatkar, Aarti论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USA AstraZeneca, R&D, Discovery Sci, Discovery Biol, Waltham, MA 02451 USA
- [5] Therapeutic potential of MCC950, a specific inhibitor of NLRP3 inflammasomeEUROPEAN JOURNAL OF PHARMACOLOGY, 2022, 928Li, Hao论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R ChinaGuan, Yanling论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R ChinaLiang, Bo论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Affiliated Hosp 1, Inst Dermatol, 81 Meishan Rd, Hefei 230032, Anhui, Peoples R China Anhui Med Univ, Affiliated Hosp 1, Dept Dermatol, 81 Meishan Rd, Hefei 230032, Anhui, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R ChinaDing, Peng论文数: 0 引用数: 0 h-index: 0机构: MOE, Key Lab Populat Hlth Life Cycle, Hefei 230032, Anhui, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R ChinaHou, Xin论文数: 0 引用数: 0 h-index: 0机构: Ningbo Univ, Sch Med, Ningbo, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R ChinaWei, Wei论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Key Lab Antiinflammatory & Immune Med, Minist Educ, Meishan Rd 81, Hefei 230032, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R ChinaMa, Yang论文数: 0 引用数: 0 h-index: 0机构: Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Key Lab Antiinflammatory & Immune Med, Minist Educ, Meishan Rd 81, Hefei 230032, Peoples R China Anhui Med Univ, Inst Clin Pharmacol, Anhui Collaborat Innovat Ctr Antiinflammatory & Im, Key Lab Antiinflammatory & Immune Med,Minist Educ, Hefei, Peoples R China
- [6] Target of MCC950 in Inhibition of NLRP3 Inflammasome Activation: a Literature ReviewINFLAMMATION, 2020, 43 (01) : 17 - 23Wu, Danbin论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaChen, Yefei论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaSun, Yingxin论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaGao, Qing论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaLi, Huhu论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaYang, Zhengfei论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaWang, Yangxue论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaJiang, Xijuan论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R ChinaYu, Bin论文数: 0 引用数: 0 h-index: 0机构: Tianjin Univ Tradit Chinese Med, Int Exchanges Dept, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Int Educ Coll, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China Tianjin Univ Tradit Chinese Med, Sch Integrat Med, 10 Poyanghu Rd,West Area, Tianjin 301617, Peoples R China
- [7] Target of MCC950 in Inhibition of NLRP3 Inflammasome Activation: a Literature ReviewInflammation, 2020, 43 : 17 - 23Danbin Wu论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineYefei Chen论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineYingxin Sun论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineQing Gao论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineHuhu Li论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineZhengfei Yang论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineYangxue Wang论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineXijuan Jiang论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative MedicineBin Yu论文数: 0 引用数: 0 h-index: 0机构: Tianjin University of Traditional Chinese Medicine,School of Integrative Medicine
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- [10] MCC950 is a potent and specific inhibitor of the NLRP3 inflammasome and a novel potential therapeutic for NLRP3 driven diseasesCYTOKINE, 2014, 70 (01) : 35 - 35Coll, Rebecca C.论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Inst Mol Biosci, Brisbane, Qld, Australia Univ Dublin Trinity Coll, Trinity Biomed Sci Inst, Dublin 2, Ireland Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaRobertson, Avril A. B.论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Inst Mol Biosci, Brisbane, Qld, Australia Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaChae, Jae Jin论文数: 0 引用数: 0 h-index: 0机构: NHGRI, Inflammatory Dis Sect, Med Genet Branch, NIH, Bethesda, MD 20892 USA Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaHiggins, Sarah C.论文数: 0 引用数: 0 h-index: 0机构: Univ Dublin Trinity Coll, Trinity Biomed Sci Inst, Dublin 2, Ireland Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaDungan, Lara S.论文数: 0 引用数: 0 h-index: 0机构: Univ Dublin Trinity Coll, Trinity Biomed Sci Inst, Dublin 2, Ireland Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaMunoz-Planillo, Raul论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Sch Med, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Sch Med, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaMonks, Brian G.论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Innate Immun, Bonn, Germany Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaCroker, Daniel E.论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Inst Mol Biosci, Brisbane, Qld, Australia Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaSutton, Caroline E.论文数: 0 引用数: 0 h-index: 0机构: Univ Dublin Trinity Coll, Trinity Biomed Sci Inst, Dublin 2, Ireland Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaStutz, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Innate Immun, Bonn, Germany Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaNunez, Gabriel论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Sch Med, Dept Pathol, Ann Arbor, MI 48109 USA Univ Michigan, Sch Med, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaLatz, Eicke论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Innate Immun, Bonn, Germany Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaKastner, Daniel L.论文数: 0 引用数: 0 h-index: 0机构: NHGRI, Inflammatory Dis Sect, Med Genet Branch, NIH, Bethesda, MD 20892 USA Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaMills, Kingston H. G.论文数: 0 引用数: 0 h-index: 0机构: Univ Dublin Trinity Coll, Trinity Biomed Sci Inst, Dublin 2, Ireland Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaMasters, Seth L.论文数: 0 引用数: 0 h-index: 0机构: Walter & Eliza Hall Inst Med Res, Melbourne, Vic 3050, Australia Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaSchroder, Kate论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Inst Mol Biosci, Brisbane, Qld, Australia Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaCooper, Matt A.论文数: 0 引用数: 0 h-index: 0机构: Univ Queensland, Inst Mol Biosci, Brisbane, Qld, Australia Univ Queensland, Inst Mol Biosci, Brisbane, Qld, AustraliaO'Neill, Luke A. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Dublin Trinity Coll, Trinity Biomed Sci Inst, Dublin 2, Ireland Univ Queensland, Inst Mol Biosci, Brisbane, Qld, Australia