A Synthesis of Tritium-Labeled Olanzapine

被引:0
|
作者
V. P. Shevchenko
I. Yu. Nagaev
Yu. V. Kuznetsov
E. V. Polunin
A. A. Zozulya
N. F. Myasoedov
机构
[1] Russian Academy of Sciences,Institute of Molecular Genetics
来源
Russian Journal of Bioorganic Chemistry | 2005年 / 31卷
关键词
olanzapine; synthesis; tritium;
D O I
暂无
中图分类号
学科分类号
摘要
A synthesis of olanzapine, 2-methyl-10-(4-methyl-1-piperazinyl)-4H-thieno[2,3-b][1,5]benzodiazepine, was carried out and the conditions for its tritium labeling were optimized to obtain a tritium-labeled olanzapine preparation with a specific radioactivity of 12 Ci/mmol.
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页码:378 / 382
页数:4
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