Multiple PIK3CA mutation clonality correlates with outcomes in taselisib + fulvestrant-treated ER+/HER2–, PIK3CA-mutated breast cancers

被引:0
作者
Katherine E. Hutchinson
Jessica W. Chen
Heidi M. Savage
Thomas J. Stout
Frauke Schimmoller
Javier Cortés
Susan Dent
Nadia Harbeck
William Jacot
Ian Krop
Sally E. Trabucco
Smruthy Sivakumar
Ethan S. Sokol
Timothy R. Wilson
机构
[1] Oncology Biomarker Development,Product Development Oncology
[2] Genentech,Department of Medicine, Faculty of Biomedical and Health Sciences
[3] Inc.,Duke Cancer Institute
[4] Genentech,Breast Center, Department Gynecology and Obstetrics and Comprehensive Cancer Center (CCC) Munich
[5] Inc.,Institut du Cancer de Montpellier (ICM) Val d’Aurelle
[6] International Breast Cancer Center (IBCC),undefined
[7] Pangaea Oncology,undefined
[8] Quironsalud Group,undefined
[9] Universidad Europea de Madrid,undefined
[10] Duke University,undefined
[11] Ludwig-Maximilians-University (LMU) Hospital,undefined
[12] Montpellier University,undefined
[13] Yale Cancer Center,undefined
[14] Foundation Medicine,undefined
[15] Inc,undefined
来源
Genome Medicine | / 15卷
关键词
Double ; mutation; Clonal; Taselisib; PI3K inhibitor; Breast cancer; ctDNA; PI3K signaling;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
相关论文
共 255 条
[1]  
Fruman DA(2017)The PI3K pathway in human disease Cell 170 605-635
[2]  
Chiu H(2004)High frequency of mutations of the PIK3CA gene in human cancers Science 304 554-713
[3]  
Hopkins BD(2017)Mutational landscape of metastatic cancer revealed from prospective clinical sequencing of 10,000 patients Nat Med 23 703-832 e823
[4]  
Bagrodia S(2017)A Pan-Cancer Proteogenomic Atlas of PI3K/AKT/mTOR pathway alterations Cancer Cell 31 820-775
[5]  
Cantley LC(2004)The PIK3CA gene is mutated with high frequency in human breast cancers Cancer Biol Ther 3 772-438 e426
[6]  
Abraham RT(2018)The genomic landscape of endocrine-resistant advanced breast cancers Cancer Cell 34 427-11000
[7]  
Samuels Y(2005)Breast cancer-associated PIK3CA mutations are oncogenic in mammary epithelial cells Cancer Res 65 10992-807
[8]  
Wang Z(2005)Phosphatidylinositol 3-kinase mutations identified in human cancer are oncogenic Proc Natl Acad Sci U S A 102 802-916
[9]  
Bardelli A(2017)Buparlisib plus fulvestrant versus placebo plus fulvestrant in postmenopausal, hormone receptor-positive, HER2-negative, advanced breast cancer (BELLE-2): a randomised, double-blind, placebo-controlled, phase 3 trial Lancet Oncol 18 904-100
[10]  
Silliman N(2018)Buparlisib plus fulvestrant in postmenopausal women with hormone-receptor-positive, HER2-negative, advanced breast cancer progressing on or after mTOR inhibition (BELLE-3): a randomised, double-blind, placebo-controlled, phase 3 trial Lancet Oncol 19 87-1668