Ankylosing spondylitis PET imaging and quantifications via P2X7 receptor-targeting radioligand [18F]GSK1482160

被引:0
|
作者
Shiyanjin Zhang
Yifan Qiu
Lihua Huang
Lei Bi
Yuanqing Guo
Ke You
Guolong Huang
Yuhan Wang
Hai Lu
Hongjun Jin
Hong Shan
机构
[1] Sun Yat-Sen University Fifth Affiliated Hospital,Department of Spine Surgery
[2] The Fifth Affiliated Hospital,Guangdong Provincial Engineering Research Center of Molecular Imaging
[3] Sun Yat-Sen University,undefined
关键词
Micro-PET/CT; Ankylosing spondylitis (AS); P2X7R; Macrophage;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:3589 / 3601
页数:12
相关论文
共 50 条
  • [1] Ankylosing spondylitis PET imaging and quantifications via P2X7 receptor-targeting radioligand [18F]GSK1482160
    Zhang, Shiyanjin
    Qiu, Yifan
    Huang, Lihua
    Bi, Lei
    Guo, Yuanqing
    You, Ke
    Huang, Guolong
    Wang, Yuhan
    Lu, Hai
    Jin, Hongjun
    Shan, Hong
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2023, 50 (12) : 3589 - 3601
  • [2] P2X7 receptor-targeting radioligand [18F]F-PTTP longitudinal pilot PET imaging in epileptic rat models
    Fu, Wenhui
    Lin, Qingyu
    Fu Zhequan
    Shi, Dai
    Yang, Tingting
    Cheng, Dengfeng
    JOURNAL OF NUCLEAR MEDICINE, 2024, 65
  • [3] Synthesis of [11C]GSK1482160 as a new PET agent for targeting P2X7 receptor
    Gao, Mingzhang
    Wang, Min
    Green, Mark A.
    Hutchins, Gary D.
    Zheng, Qi-Huang
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (09) : 1965 - 1970
  • [4] Synthesis of [11C]GSK1482160 as a potential PET agent for imaging of P2X7 receptor
    Gao, Mingzhang
    Zheng, Qi-Huang
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248
  • [5] Synthesis of [11C] GSK1482160 as a new potential PET radiopharmaceutical for targeting the P2X7 receptor
    Gao, Mingzhang
    Wang, Min
    Green, Mark
    Hutchins, Gary
    Zheng, Qi-Huang
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2015, 58 : S273 - S273
  • [6] Initial characterization of [11C]-GSK1482160 as radioligand for P2X7 receptors
    Meyer, Jill
    Peters, Jonathan
    Riley, Amanda
    McCarthy, Brian
    Gao, Minzhang
    Wang, Min
    Zheng, Qi-Huang
    Hutchins, Gary
    Territo, Paul
    JOURNAL OF NUCLEAR MEDICINE, 2016, 57
  • [7] Pharmacologic characterizations of a P2X7 receptor-specific radioligand, [11C]GSK1482160 for neuroinflammatory response
    Han, Junbin
    Liu, Hui
    Liu, Chunling
    Jin, Hongjun
    Perlmutter, Joel S.
    Egan, Terrance M.
    Tu, Zhude
    NUCLEAR MEDICINE COMMUNICATIONS, 2017, 38 (05) : 372 - 382
  • [8] Increased Cerebral Level of P2X7R in a Tauopathy Mouse Model by PET Using [18F]GSK1482160
    Kong, Yanyan
    Cao, Lei
    Wang, Jiao
    Zhuang, Junyi
    Liu, Yongshan
    Bi, Lei
    Qiu, Yifan
    Hou, Yuyi
    Huang, Qi
    Xie, Fang
    Yang, Yunhao
    Shi, Kuangyu
    Rominger, Axel
    Guan, Yihui
    Jin, Hongjun
    Ni, Ruiqing
    ACS CHEMICAL NEUROSCIENCE, 2024, 15 (11): : 2112 - 2120
  • [9] Radiosynthesis of P2X7 receptor radioligands [11C]GSK1482160 and [11C]GSK1482160 isomer under different base conditions
    Gao, Mingzhang
    Wang, Min
    Zheng, Qi-Huang
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253
  • [10] Development and Validation of HPLC Methods for Determination and Analysis of [11C]GSK1482160, a Radiopharmaceutical for Targeting the P2X7 Receptor
    Wissmann, Carmen
    Wang, Min
    Gao, Mingzhang
    Zheng, Qihuang
    Glick-Wilson, Barbara
    Green, Mark
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2017, 60 : S571 - S571