Microwave assisted selective synthesis of (E)-1-(4-Chloro-7-hydroxy-2-aryl-2H-chromen-6-yl)-3-arylprop-2-en-1-ones and their antimicrobial activity

被引：0
作者：
D. Ashok
M. Sarasija
D. Shravani
B. Vijayalaxmi
K. Sudershan
机构：
[1] Osmania University,Green and Medicinal Chemistry Laboratory, Department of Chemistry
来源：
Russian Journal of General Chemistry | 2016年 / 86卷
关键词：
chlorochromene frame work; selective cyclization; microwave irradiation; antimicrobial activity;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
A series of new (E)-1-(4-chloro-7-hydroxy-2-aryl-2H-chromen-6-yl)-3-arylprop-2-en-1-ones (2a–2f) have been synthesized by selective mono cyclization of 4,6-dicinnamoyl resorcinols (1a–1f) using Vilsmeier–Haack reagent under conventional heating and microwave irradiation. The structures of the synthesized compounds have been elucidated by elemental analysis, IR, 1H NMR, 13C NMR and Mass spectral data. The synthesized compounds were tested in vitro for antimicrobial activity.
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页码：930 / 933
页数：3
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