4-aroylpiperidines and 4-(α-hydroxyphenyl)piperidines as selective sigma-1 receptor ligands: synthesis, preliminary pharmacological evaluation and computational studies

被引:0
作者
Hermia N. Ikome
Fidele Ntie-Kang
Moses N. Ngemenya
Zhude Tu
Robert H. Mach
Simon M. N. Efange
机构
[1] University of Buea,Department of Chemistry, Faculty of Science
[2] Martin-Luther University of Halle-Wittenberg,Department of Pharmaceutical Chemistry
[3] University of Buea,Biotechnology Unit, Department of Biochemistry and Molecular Biology, Faculty of Science
[4] University of Washington School of Medicine,Department of Radiology
来源
Chemistry Central Journal | / 10卷
关键词
Sigma-1 binding; Piperidines; QSAR; Pharmacophore;
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