Synthesis, structure, and antimicrobial activity of methyl (4-alkanoyl-3-hydroxy-1,5-diaryl-1H-pyrrol-2-yl)acetates

被引：0
|
作者：
P. P. Mukovoz
P. A. Slepukhin
O. S. El’tsov
I. N. Ganebnykh
A. V. Gorbunova
A. N. Sizentsov
M. L. Rusyaeva
机构：
[1] Moscow Institute of Technology (Orenburg Branch),
[2] Postovskii Institute of Organic Synthesis,undefined
[3] Yeltsin Ural Federal University,undefined
[4] Orenburg State University,undefined
来源：
Russian Journal of General Chemistry | 2017年 / 87卷
关键词：
3,4-dihydroxy-6-oxo-2,4-alkadienoic acids esters; arylidenearylamines; (4-alkanoyl-3-hydroxy-1,5-diaryl-1; -pyrrol-2-yl)acetic acids esters;
D O I：
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学科分类号：
摘要：
Reactions of methyl 3,4,6-trioxoalkanoates (3,4-dihydroxy-6-oxo-2,4-alkadienoates) with a mixture of arylamines and aromatic aldehydes or with the corresponding arylidenearylamines lead to the formation of methyl (4- alkanoyl-3-hydroxy-1,5-diaryl-1H-pyrrol-2-yl)acetates. Structure of the synthesized compounds is discussed basing on IR, 1H NMR spectroscopy, mass spectrometry, and X-ray diffraction data.
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页码：2291 / 2298
页数：7
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