One-pot multicomponent synthesis of two novel thiolactone scaffolds

被引：0
|
作者：
B. Beck
S. Srivastava
K. Khoury
E. Herdtweck
Alexander Dömling
机构：
[1] University of Pittsburgh,Department of Pharmacy
[2] Technical University Munich,undefined
来源：
Molecular Diversity | 2010年 / 14卷
关键词：
Multicomponent reaction (MCR); Isocyanide; Thiolactone; Virtual library;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
We designed two novel thiolactone scaffolds. Both scaffolds can be accessed by a convergent Ugi multicomponent reaction (MCR) and are, thus, amenable to library synthesis. Design, stereoselectivity, structures, full experimental details, and virtual libraries will be reported.
引用
收藏
页码：479 / 491
页数：12
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