Synthesis, structure, and antimicrobial activity of methyl (4-alkanoyl-1,5-diaryl-2-hydroxy-3-oxo-2,3-dihydro-1H-pyrrol-2-yl)acetates

被引：0

作者：

P. P. Mukovoz

A. V. Gorbunova

P. A. Slepukhin

O. S. El’tsov

I. N. Ganebnykh

A. N. Sizentsov

I. V. Korobova

机构：

[1] Moscow Institute of Technology,Orenburg Branch

[2] Orenburg State University,Postovskii Institute of Organic Synthesis, Ural Branch

[3] Russian Academy of Sciences,undefined

[4] Yeltsin Ural Federal University,undefined

来源：

Russian Journal of General Chemistry | 2017年 / 87卷

关键词：

3,4-dihydroxy-6-oxo-2,4-alkadienoic acid esters; (4-alkanoyl-1,5-diaryl-2-hydroxy-3-oxo-2,3-dihydro-1; -pyrrol-2-yl)acetic acid esters; 1,3,4,6-tetracarbonyl compounds;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

Reactions of methyl 3,4,6-trioxoalkanoates (3,4-dihydroxy-6-oxo-2,4-alkadienoates) with mixtures of aromatic aldehydes and arylamines or with the corresponding N-(arylmethylidene)anilines afforded methyl (4-alkanoyl-1,5-diaryl-2-hydroxy-3-oxo-2,3-dihydro-1H-pyrrol-2-yl)acetates. The product structure was discussed on the basis of their IR, 1H NMR, and mass spectra and X-ray diffraction data, and their antimicrobial activity against Staphylococcus aureus P-209 and Escherichia coli M17 was evaluated.

引用

页码：1695 / 1701

页数：6

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