3-Chlorophenylboronic acid-promoted, one-pot, aza-Friedel–Crafts reaction of indoles

被引：0
作者：
Santosh V. Goswami
Prashant B. Thorat
Mahesh V. Shukla
Sudhakar R. Bhusare
机构：
[1] Dnyanopasak College,Department of Chemistry
来源：
Research on Chemical Intermediates | 2015年 / 41卷
关键词：
Aza-Friedel–Crafts reaction; 3-Chlorophenylboronic acid; Indole; Aromatic aldehyde; ,; -Dimethylaniline;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
3-Chlorophenylboronic acid promotes efficient synthesis of 3-substituted indole derivatives via aza-Friedel–Crafts reaction of indoles, aromatic aldehydes, and N,N-dimethylaniline at room temperature. The mild reaction conditions, excellent yields, and easy experimental workup are striking features of this procedure for synthesis of 3-substituted indoles.
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页码：2583 / 2589
页数：6
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