Some chemical properties of 2,3-dihydro-4H-[1,3]thiazino[3,2-a] benzimidazol-4-one and 2-aryl-2,3-dihydro-4H-[1,3]thiazino[3,2-a]benzimidazol-4- ones

被引:0
作者
Britsun V.N. [1 ]
Esipenko A.N. [1 ]
Lozinskii M.O. [1 ]
机构
[1] Institute of Organic Chemistry, National Academy of Sciences of Ukraine
来源
Chem. Heterocycl. Compd. | 2006年 / 3卷 / 396-402期
关键词
2,3-dihydro-4H-[1,3]-thiazino[3,2-a]benzimidazol-4-one; 2-aryl-2,3-dihydro-4H-[1,3]thiazino[3,2-a]benzimidazol-4-ones; Alkylation; Amination; Oxidation;
D O I
10.1007/s10593-006-0099-x
中图分类号
学科分类号
摘要
We have studied the reaction of 2,3-dihydro-4H-[1,3]thiazino[3,2-a] benzimidazol-4-one and 2-aryl-2,3-dihydro-4H-[1,3]thiazino[3,2-a]benzimidazol-4- ones with amines, alkylating reagents, and hydrogen peroxide. We have shown that the presence of an aryl substituent at the 2 position of [1,3-thiazino[3,2-a] benzimidazol-4-ones has a substantial effect on the direction of the reactions. ©2006 Springer Science+Business Media, Inc.
引用
收藏
页码:396 / 402
页数:6
相关论文
共 50 条
  • [31] Biomimetic hydrogenation of electron deficient olefins using in situ generated 2-arylbenzimidazoline: synthesis of novel 3-benzylbenzo[4,5]thiazolo[3,2-a]pyrimidin-4-ones
    Danehchin, Maryam
    Esmaeili, Abbas Ali
    MOLECULAR DIVERSITY, 2022, 26 (02) : 1191 - 1199
  • [32] (4Z)-1-Benzyl(1,3-Dibenzyl)-4-(2-oxopropylidene)-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-2-one
    Said, Ould Mohamed Sidya Mohamed
    Rachid, Bouhfid
    Joly, Nicolas
    Lequart, Vincent
    Martin, Patrick
    Massoui, M.
    Essassi, El Mokhtar
    MOLBANK, 2006, (05)
  • [33] (4Z)-1-Propargyl(1,3-Dipropargyl)-4-(2-oxopropylidene)-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-2-one
    Said, Ould Mohamed Sidya Mohamed
    Rachid, Bouhfid
    Joly, Nicolas
    Lequart, Vincent
    Martin, Patrick
    Massoui, M.
    Essassi, El Mokhtar
    MOLBANK, 2006, (05)
  • [34] Cross-dehydrogenative coupling of 3,6-dihydro-2H-pyrans with 1,3-dicarbonyls and aryl moieties
    Feng, Guidong
    Sun, Chuanxi
    Xin, Xiaodong
    Wan, Renzhong
    Liu, Lei
    TETRAHEDRON LETTERS, 2019, 60 (23) : 1547 - 1550
  • [35] Synthesis and antibacterial activity of some new 2,3-dimethoxy-3-hydroxy-2-(1-phenyl-3-aryl-4-pyrazolyl)chromanones
    Prakash, Om
    Kumar, Rajesh
    Sehrawat, Rakesh
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2009, 44 (04) : 1763 - 1767
  • [36] Synthesis of 1H-pyrano[4,3-b]benzofuran-1-one derivatives via photochemical cyclization of substituted 4H-furo[3,2-c]pyran-4-ones
    Milyutin, Constantine, V
    Lichitsky, Boris, V
    Melekhina, Valeriya G.
    Komogortsev, Andrey N.
    Fakhrutdinov, Artem N.
    Minyaev, Mikhail E.
    Krayushkin, Michail M.
    TETRAHEDRON LETTERS, 2020, 61 (44)
  • [37] Sequential Ugi Four-Component Reaction (4-CR)/C-H Activation Using (Diacetoxyiodo)benzene for the Synthesis of 3-(Diphenylmethylidene)-2,3-dihydro-1H-indol-2-ones
    Ghabraie, Elmira
    Balalaie, Saeed
    HELVETICA CHIMICA ACTA, 2014, 97 (11) : 1555 - 1563
  • [38] 3,4-Dihydro-3H-pyrrol-2-imines as Conformationally Restrained 1,3-Diazabutadienes: Synthesis, Structural Properties and Protonation
    Janich, Simon
    Froehlich, Roland
    Wilken, Andrea
    von Zamory, Jan
    Wakamiya, Atsushi
    Yamaguchi, Shigehiro
    Wuerthwein, Ernst-Ulrich
    EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2009, 2009 (13) : 2077 - 2087
  • [39] 2-(2-Chloro-6,7-dimethylquinolin-3-yl)-2,3-dihydroquinolin-4(1H)-one
    Benzerka, Saida
    Bouraiou, Abdelmalek
    Bouacida, Sofiane
    Roisnel, Thierry
    Belfaitah, Ali
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2011, 67 : O2084 - U949
  • [40] One-Pot Multicomponent Synthesis of Pyrrolo[1,2-a]pyrazines in Water Catalyzed by Fe3O4@SiO2-OSO3H
    Rostami, Hedieh
    Shiri, Lotfi
    CHEMISTRYSELECT, 2018, 3 (47): : 13487 - 13492