Inhibition Requirements of the Human Apical Sodium-Dependent Bile Acid Transporter (hASBT) Using Aminopiperidine Conjugates of glutamyl-Bile Acids

被引:0
作者
Pablo M. González
Chayan Acharya
Alexander D. MacKerell
James E. Polli
机构
[1] University of Maryland,Department of Pharmaceutical Sciences, School of Pharmacy
[2] Pontificia Universidad Católica de Chile,Departamento de Farmacia, Facultad de Química
来源
Pharmaceutical Research | 2009年 / 26卷
关键词
apical sodium-dependent bile acid transporter; bile acid; CHARMM; conformationally sampled pharmacophore; transporter;
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页码:1665 / 1678
页数:13
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