Novel convenient one-pot method for the synthesis of indoloquinolines

被引:0
作者
N. A. Aksenov
A. Z. Gasanova
G. M. Abakarov
I. V. Aksenova
A. V. Aksenov
机构
[1] North Caucasus Federal University,
[2] Dagestan State Technical University,undefined
来源
Russian Chemical Bulletin | 2019年 / 68卷
关键词
Fischer indole synthesis; isocryptolepine; reduction; synthesis; indole;
D O I
暂无
中图分类号
学科分类号
摘要
A novel one-pot method based on the sequence of the Fisher reaction between nitroacetophenone and phenylhydrazines, the reduction with metallic tin directly in polyphosphoric acid, and acylation has been developed for the synthesis of indoloquinolines. The obtained indolo-[3,2-c]quinolines are precursors of the analogs of isocryptolepine alkaloid.
引用
收藏
页码:836 / 840
页数:4
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